| Identification | Back Directory | [Name]
6-[5-[(2S)-2-AZETIDINYLMETHOXY]-3-PYRIDINYL]-5-HEXYN-1-OL DIHYDROCHLORIDE | [CAS]
820231-95-6 | [Synonyms]
Sazetidine A
SAZETIDINE A DIHYDROCHLORIDE
(S)-6-(5-(azetidin-2-ylmethoxy)pyridin-3-yl)hex-5-yn-1-ol
5-Hexyn-1-ol, 6-[5-[(2S)-2-azetidinylmethoxy]-3-pyridinyl]-
6-[5-[[(2S)-azetidin-2-yl]methoxy]pyridin-3-yl]hex-5-yn-1-ol
6-[5-[(2S)-2-AZETIDINYLMETHOXY]-3-PYRIDINYL]-5-HEXYN-1-OL DIHYDROCHLORIDE | [Molecular Formula]
C15H20N2O2 | [MDL Number]
MFCD09971128 | [MOL File]
820231-95-6.mol | [Molecular Weight]
260.33 |
| Hazard Information | Back Directory | [Biological Activity]
Subtype-selective α 4 β 2 nicotinic acetylcholine receptor ligand (K i values are 0.26 and 54 nM at α 4 β 2 and α 3 β 4 receptors respectively). May act as a silent desensitizer or as an agonist (EC 50 = 1.1 nM for nAChR-stimulated dopamine release). Exhibits analgesic activity in vivo . |
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