Furin Inhibitor II - Calbiochem

Furin Inhibitor II - Calbiochem Struktur
CAS-Nr.
Englisch Name:
Furin Inhibitor II - Calbiochem
Synonyma:
Furin Inhibitor II - Calbiochem
CBNumber:
CB74817205
Summenformel:
Molgewicht:
0
MOL-Datei:
Mol file

Furin Inhibitor II - Calbiochem Eigenschaften

Sicherheit

Furin Inhibitor II - Calbiochem Chemische Eigenschaften,Einsatz,Produktion Methoden

Allgemeine Beschreibung

A polyarginine compound that acts as a potent, specific, and competitive inhibitor of furin (Ki = 106 nM). Inhibits Subtilisin-like proprotein convertase 4 (PACE4) and prohormone convertase 1 (PC1) at much higher concentration (Ki = 580 nM and 13 μM, respectively). Has a stimulatory effect on the activity of prohormone convertase 2 (PC2). The D-peptides are suggested to be more resistant to in vivo hydrolysis than L-peptides.

Biochem/physiol Actions

Primary Targetfurin

Furin Inhibitor II - Calbiochem Upstream-Materialien And Downstream Produkte

Upstream-Materialien

Downstream Produkte


Furin Inhibitor II - Calbiochem Anbieter Lieferant Produzent Hersteller Vertrieb Händler.

Global( 2)Lieferanten
Firmenname Telefon E-Mail Land Produktkatalog Edge Rate
Sigma-Aldrich 021-61415566 800-8193336
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