UFP-101
- CAS No.
- 849024-68-6
- Chemical Name:
- UFP-101
- Synonyms
- UFP-101;PubChem ID: 16152632;[NPHE1, ARG14, LYS15]NOCICEPTIN-NH2;N-(BZL)GLY-GLY-GLY-PHE-THR-GLY-ALA-ARG-LYS-SER-ALA-ARG-LYS-ARG-LYS-ASN-GLN-NH2;N-(Bzl)Gly-Gly-Gly-Phe-Thr-Gly-Ala-Arg-Lys-Ser-Ala-Arg-Lys-Arg-Lys-Asn-Gln-NH2 (N-(Bzl)GlyN-Benzylglycine);L-Glutamamide, N-(phenylmethyl)glycylglycylglycyl-L-phenylalanyl-L-threonylglycyl-L-alanyl-L-arginyl-L-lysyl-L-seryl-L-alanyl-L-arginyl-L-lysyl-L-arginyl-L-lysyl-L-asparaginyl- (9CI)
- CBNumber:
- CB4763828
- Molecular Formula:
- C82H138N32O21
- Molecular Weight:
- 1908.17
- MDL Number:
- MFCD04112664
- MOL File:
- Mol file
- MSDS File:
- SDS
- TDS File:
- TDS
| Product description | Number | Pack Size | Price |
| UFP-101 | 1552 | 1 | $364 |
| UFP-101 | B5128 | 1mg | $534 |
| UFP-101 95.00% | BRS0000791 | 0.5MG | $684.92 |
| UFP-101 95.00% | BRS0000791 | 1MG | $846.5 |
| UFP-101 95.00% | BRS0000791 | 5MG | $1829.52 |
UFP-101 price More Price(5)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Tocris | 1552 | UFP-101 | 849024-68-6 | 1 | $364 | 2021-12-16 | Buy |
| ApexBio Technology | B5128 | UFP-101 | 849024-68-6 | 1mg | $534 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | BRS0000791 | UFP-101 95.00% | 849024-68-6 | 0.5MG | $684.92 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | BRS0000791 | UFP-101 95.00% | 849024-68-6 | 1MG | $846.5 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | BRS0000791 | UFP-101 95.00% | 849024-68-6 | 5MG | $1829.52 | 2021-12-16 | Buy |
UFP-101 Chemical Properties,Uses,Production
Uses
UFP-101 is a potent, selective, and competitive antagonist of the NOP receptor, with a pKi of 10.24. UFP-101 displays >3000-fold selectivity over δ, μ and κ opioid receptors. UFP-101 shows antidepressant-like effect[1][2].
in vivo
UFP-101 elicits a pronounced acute and dosedependent antidepressant-like effect in mice submitted to the forced swimming test (FST)[1].
IC 50
NOP Receptor/ORL1
storage
Store at -20°C
References
[1] Calo G, et al. [Nphe1,Arg14,Lys15]nociceptin-NH2, a novel potent and selective antagonist of the nociceptin/orphanin FQ receptor. Br J Pharmacol. 2002;136(2):303-311. DOI:10.1038/sj.bjp.0704706
[2] Gavioli EC, et al. Blockade of nociceptin/orphanin FQ-NOP receptor signalling produces antidepressant-like effects: pharmacological and genetic evidences from the mouse forced swimming test. Eur J Neurosci. 2003;17(9):1987-1990. DOI:10.1046/j.1460-9568.2003.02603.x
UFP-101 Preparation Products And Raw materials
Raw materials
Preparation Products
UFP-101 Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Shenzhen Nexconn Pharmatechs Ltd | +86-755-89396905 +86-15013857715 | admin@nexconn.com | China | 10404 | 58 |
| BOC Sciences | +1-631-485-4226 | inquiry@bocsci.com | United States | 19552 | 58 |
| Career Henan Chemica Co | +86-0371-86658258 +8613203830695 | laboratory@coreychem.com | China | 30227 | 58 |
| Zhejiang J&C Biological Technology Co.,Limited | +1-2135480471 +1-2135480471; | sales@sarms4muscle.com | China | 10473 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 57505 | 58 | |
| Changsha MOL Changes Biotechnology Co., Ltd. | +8619375158599 | info@molchanges.com | China | 5218 | 58 |
| 3B Pharmachem (Wuhan) International Co.,Ltd. | 821-50328103-801 18930552037 | 3bsc@sina.com | China | 15838 | 69 |
| Chemsky（shanghai）International Co.,Ltd. | 021-50135380 | shchemsky@sina.com | China | 32321 | 50 |
| Hunan Hui Bai Shi Biotechnology Co., Ltd. | 0731-85526065 13308475853 | ivy@hnhbsj.com | China | 7245 | 62 |
| Creative Peptides | info@creative-peptides.com | United States | 6083 | 56 |
