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AS-1763

CAS No.
2227211-00-7
Chemical Name:
AS-1763
Synonyms
AS-1763;Milrebrutinib
CBNumber:
CB710270933
Molecular Formula:
C33H31FN6O3
Molecular Weight:
578.65
MDL Number:
MOL File:
2227211-00-7.mol
Last updated:2023-05-09 09:30:48

AS-1763 Properties

FDA UNII 4E4EWP9DJQ

AS-1763 Chemical Properties,Uses,Production

Biological Activity

AS-1763 is a potent, selective, noncovalent, and orally available inhibitor of Bruton’s tyrosine kinase (IC50 = 0.85 nM).

References

[1]. Kawahata W, et al. Discovery of AS-1763: A Potent, Selective, Noncovalent, and Orally Available Inhibitor of Bruton’s Tyrosine Kinase. J Med Chem. 2021 Oct 14;64(19):14129-14141.

AS-1763 Preparation Products And Raw materials

Raw materials

Preparation Products

AS-1763 Suppliers

Global( 9)Suppliers
Supplier Tel Email Country ProdList Advantage
ShangHai Caerulum Pharma Discovery Co., Ltd. 18149758185 sales-cpd@caerulumpharma.com China 3423 58
Shanghai XingMo Biotechnology Co., Ltd. 13524779951 2075692521@qq.com China 309 55
Shanghai Chaolan Chemical Technology Center QQ:65489617 15618227136 info@SuperLan-chem.com China 9779 58
Heze Development Zone chuangli Chemical Co., Ltd. +86-530-529 6766,+86-15666160102 15666160102 info@chuangli-chem.com China 876 55
DC Chemicals 021-58447131 13564518121 sales@dcchemicals.com China 9414 58
Suzhou youruike Chemical Pharmaceutical Technology Co., Ltd 15317229551 15151849396@163.com China 997 58
Chunchuang (Wuhan) Technology Co., Ltd 15342225168 yutianchun2007@126.com China 10006 58
Hebei Weite Medical Technology Co., Ltd 13180081292 contact@wetogethermed.com China 7304 58
Wuhan Shanhai Zhihe Biotechnology Co., Ltd. 17771424646 shoubull@126.com China 966 58
AS-1763 Milrebrutinib 2227211-00-7