PD144418 OXALATE 化学特性,用途語,生産方法
用途
高親和性で選択的 σ1 リガンドです(Ki = 0.08 nM(σ1),1377 nM(σ2)。
用途
高親和性で選択的 σ1 リガンドです(Ki = 0.08 nmol/l(σ1),1,377 nmol/l(σ2))。
使用
PD 144418 is high affinity, selective σ1 ligand (Ki values are 0.08 and 1377 nM for σ1 and σ2 respectively). PD 144418 displays no significant activity at a wide range of other receptors, ion channels and enzymes. PD 144418 antagonizes mescaline-induced scratching in mice following i.p. administration.
生物活性
High affinity, selective σ 1 ligand (K i values are 0.08 and 1377 nM for σ 1 and σ 2 respectively). Displays no significant activity at a wide range of other receptors, ion channels and enzymes. Antagonizes mescaline-induced scratching in mice following i.p. administration.
PD144418 OXALATE 上流と下流の製品情報
原材料
準備製品