PANCREATIC POLYPEPTIDE, HUMAN

PANCREATIC POLYPEPTIDE, HUMAN 구조식 이미지
카스 번호:
75976-10-2
상품명:
PANCREATIC POLYPEPTIDE, HUMAN
동의어(영문):
PP, HUMAN;PANCREATIC POLYPEPTIDE;Human pancreatic polypeptide;PANCREATIC POLYPEPTIDE, HUMAN;M.W. 4181.71 C185H287N53O54S2;Pancreatic polypeptide(human) (9CI);PANCREATIC POLYPEPTIDE, HUMAN USP/EP/BP;APLEPVYPGDNATPEQMAQYAADLRRYINMLTRPRY-NH2;Pancreatic Polypeptide human, ≥95% (HPLC);Pancreatic Polypeptide huManPancreatic Polypeptide
CBNumber:
CB6764364
분자식:
C185H287N53O54S2
포뮬러 무게:
4181.71098
MOL 파일:
75976-10-2.mol

PANCREATIC POLYPEPTIDE, HUMAN 속성

저장 조건
-15°C
용해도
Water: 1 mg/ml
물리적 상태
가루
수용성
물에 0.70mg/ml까지 용해됨

안전

PANCREATIC POLYPEPTIDE, HUMAN C화학적 특성, 용도, 생산

개요

Pancreatic polypeptide is an agonist of neuropeptide Y (NPY) receptors that reduces forskolin-induced cAMP accumulation in L-M(TK-) cells recombinantly expressing human and rat Y4 receptors (EC50s = 87.1 and 36.3 pM, respectively). It binds to Y1 and Y5 receptors with Ki values of 19 and 3.9 nM, respectively, for human and 50 and 2.4 nM, respectively, for rhesus monkey receptors. Pancreatic polypeptide also binds to rabbit Y1, Y2, Y4, and Y5 receptors (Kis = 0.39, 0.087, 0.79, and 0.24 nM, respectively). It induces contractile responses in isolated rat colon with EC50 values of 1.6 and 0.7 nM for ascending and descending colon segments, respectively. In vivo, pancreatic polypeptide (0.7-7 nmol, i.c.v.) increases food intake in rats.

PANCREATIC POLYPEPTIDE, HUMAN 준비 용품 및 원자재

원자재

준비 용품


PANCREATIC POLYPEPTIDE, HUMAN 공급 업체

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