RILMENIDINE HEMIFUMARATE SALT
- $40 - $780
- Product name: RILMENIDINE HEMIFUMARATE SALT
- CAS: 207572-68-7
- MF: 2C10H16N2O.C4H4O4
- MW: 476.57
- EINECS:
- MDL Number:MFCD09878261
- Synonyms:RILMENIDINE HEMIFUMARATE SALT;n-(dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt;Oxaminozoline hemifumarate salt, Rilmenidene hemifumarate salt, N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt;LZFATBMLSYHRTC-WXXKFALUSA-N
12 prices
Selected condition:
Brand
- American Custom Chemicals Corporation
- ApexBio Technology
- Cayman Chemical
- ChemScene
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TRC
Package
- 1mg
- 5MG
- 10mg
- 25mg
- 50mg
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0019412
- Product descriptionRILMENIDINE HEMIFUMARATE 95.00%
- Packaging5MG
- Price$498.85
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC3965
- Product descriptionRilmenidine(hemifumarate)
- Packaging10mg
- Price$182
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number16988
- Product descriptionRilmenidine (hemifumarate) ≥98%
- Packaging1mg
- Price$40
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16988
- Product descriptionRilmenidine (hemifumarate) ≥98%
- Packaging5mg
- Price$98
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16988
- Product descriptionRilmenidine (hemifumarate) ≥98%
- Packaging10mg
- Price$161
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16988
- Product descriptionRilmenidine (hemifumarate) ≥98%
- Packaging50mg
- Price$618
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-0019424
- Product descriptionRilmenidine(hemifumarate) ≥98.0%
- Packaging5mg
- Price$375
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-0019424
- Product descriptionRilmenidine(hemifumarate) ≥98.0%
- Packaging10mg
- Price$780
- Updated2021-12-16
- Buy
- ManufacturerMedical Isotopes, Inc.
- Product number75416
- Product descriptionRilmenidine hemifumarate salt
- Packaging5mg
- Price$290
- Updated2021-12-16
- Buy
- ManufacturerSigma-Aldrich
- Product numberR134
- Product descriptionRilmenidine hemifumarate salt solid
- Packaging5mg
- Price$148
- Updated2024-03-01
- Buy
- ManufacturerSigma-Aldrich
- Product numberR134
- Product descriptionRilmenidine hemifumarate salt solid
- Packaging25mg
- Price$562
- Updated2024-03-01
- Buy
- ManufacturerTRC
- Product numberR509705
- Product descriptionRilmenidineHemifumarate
- Packaging1mg
- Price$50
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
American Custom Chemicals Corporation | API0019412 | RILMENIDINE HEMIFUMARATE 95.00% | 5MG | $498.85 | 2021-12-16 | Buy |
ApexBio Technology | C3965 | Rilmenidine(hemifumarate) | 10mg | $182 | 2021-12-16 | Buy |
Cayman Chemical | 16988 | Rilmenidine (hemifumarate) ≥98% | 1mg | $40 | 2024-03-01 | Buy |
Cayman Chemical | 16988 | Rilmenidine (hemifumarate) ≥98% | 5mg | $98 | 2024-03-01 | Buy |
Cayman Chemical | 16988 | Rilmenidine (hemifumarate) ≥98% | 10mg | $161 | 2024-03-01 | Buy |
Cayman Chemical | 16988 | Rilmenidine (hemifumarate) ≥98% | 50mg | $618 | 2024-03-01 | Buy |
ChemScene | CS-0019424 | Rilmenidine(hemifumarate) ≥98.0% | 5mg | $375 | 2021-12-16 | Buy |
ChemScene | CS-0019424 | Rilmenidine(hemifumarate) ≥98.0% | 10mg | $780 | 2021-12-16 | Buy |
Medical Isotopes, Inc. | 75416 | Rilmenidine hemifumarate salt | 5mg | $290 | 2021-12-16 | Buy |
Sigma-Aldrich | R134 | Rilmenidine hemifumarate salt solid | 5mg | $148 | 2024-03-01 | Buy |
Sigma-Aldrich | R134 | Rilmenidine hemifumarate salt solid | 25mg | $562 | 2024-03-01 | Buy |
TRC | R509705 | RilmenidineHemifumarate | 1mg | $50 | 2021-12-16 | Buy |
Properties
storage temp. :Store at -20°C
solubility :DMSO: >10mg/mL
form :solid
color :white
solubility :DMSO: >10mg/mL
form :solid
color :white
Safety Information
Symbol(GHS): | ||||||||
---|---|---|---|---|---|---|---|---|
Signal word: | ||||||||
Hazard statements: |
|
|||||||
Precautionary statements: |
|
Description
Rilmenidine is a centrally acting antihypertensive agent that has been shown to lower arterial pressure in various animal models by inhibiting the tonic activity of sympathoexcitatory neurons in the rostral ventrolateral medulla. Rilmenidine targets the nonadrenergic imidazoline-binding site I1 receptor with a Ki value of 7.1 nM and demonstrates weaker affinity for the I2 receptor with a Ki value of 5.2 μM. It can also act as an agonist of α2-adrenergic receptors, but demonstrates ~30-fold greater selectivity for I1 receptors compared to α2-adrenergic receptors. Rilmenidine is reported to induce autophagy as evidenced by a ~350% increase in LC3-II levels in PC12 cells when treated with 1 μM of the I1 agonist.Suppliers and manufacturers
Hangzhou MolCore BioPharmatech Co.,Ltd.
Shenyang Zhongshen Zekang Biomedical Technology Research Co., Ltd
Aladdin Scientific
ShangHai Caerulum Pharma Discovery Co., Ltd.
Sigma-Aldrich
Shanghai EFE Biological Technology Co., Ltd.
Shanghai Chaolan Chemical Technology Center
Beijing Jin Ming Biotechnology Co., Ltd.
BOC Sciences
ChemeGen(Shanghai) Biotechnology Co.,Ltd.