AZD3965
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- $27 - $5672
- Product name: AZD3965
- CAS: 1448671-31-5
- MF: C21H24F3N5O5S
- MW: 515.51
- EINECS:
- MDL Number:MFCD28963899
- Synonyms:5-[[(4S)-4-Hydroxy-4-methyl-2-isoxazolidinyl]carbonyl]-3-methyl-1-(1-methylethyl)-6-[[5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]methyl]-thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione;(S)-5-(4-hydroxy-4-methylisoxazolidine-2-carbonyl)-1-isopropyl-3-methyl-6-((5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)methyl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione;CS-2201;AZD-3965;AZD3965;AZD 3965;5-{[(4S)-4-Hydroxy-4-methyl-1,2-oxazolidin-2-yl]carbonyl}-1-isopropyl-3-methyl-6-{[5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]methyl}thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione;Thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione, 5-[[(4S)-4-hydroxy-4-methyl-2-isoxazolidinyl]carbonyl]-3-methyl-1-(1-methylethyl)-6-[[5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]methyl]-;AZD3965,inhibit,Inhibitor,Monocarboxylate Transporter;AZD3965, 10 mM in DMSO
47 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- ApexBio Technology
- Arctom
- Biosynth
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- TRC
Package
- 10mM*1mLinDMSO(Solid+Solvent)
- 10mM*1mLinDMSO(Solution)
- 2.5mg
- 1mg
- 2mg
- 10mM(1mLinDMSO)
- 5mg
- 10mg
- 25mg
- 50mg
- 100MG
- 200mg
- 250mg
- 1G
- Manufactureraablocks
- Product numberAA001K69
- Product descriptionAZD3965 98%
- Packaging1mg
- Price$27
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001K69
- Product descriptionAZD3965 98%
- Packaging2mg
- Price$41
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001K69
- Product descriptionAZD3965 98%
- Packaging5mg
- Price$61
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001K69
- Product descriptionAZD3965 98%
- Packaging10mg
- Price$95
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001K69
- Product descriptionAZD3965 98%
- Packaging25mg
- Price$170
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001K69
- Product descriptionAZD3965 95%
- Packaging250mg
- Price$1130
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberM22559
- Product descriptionAZD3965 98%
- Packaging1G
- Price$2450
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberM22559
- Product descriptionAZD3965 98%
- Packaging25MG
- Price$180
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberM22559
- Product descriptionAZD3965 98%
- Packaging5MG
- Price$65
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberM22559
- Product descriptionAZD3965 98%
- Packaging100MG
- Price$495
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product number7027CR
- Product descriptionCID10369242
- Packaging50mg
- Price$758
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC5049
- Product descriptionAZD 3965
- Packaging10mg
- Price$240
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberC5049
- Product descriptionAZD 3965
- Packaging25mg
- Price$430
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberC5049
- Product descriptionAZD 3965
- Packaging5mg
- Price$150
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberHY-12750
- Product descriptionAZD3965 99.93%
- Packaging10mM*1mLinDMSO(Solution)
- Price$155
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-12750
- Product descriptionAZD3965 99.93%
- Packaging10mg
- Price$171
- Updated2026-05-26
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA001K69 | AZD3965 98% | 1mg | $27 | 2026-05-28 | Buy |
| aablocks | AA001K69 | AZD3965 98% | 2mg | $41 | 2026-05-28 | Buy |
| aablocks | AA001K69 | AZD3965 98% | 5mg | $61 | 2026-05-28 | Buy |
| aablocks | AA001K69 | AZD3965 98% | 10mg | $95 | 2026-05-28 | Buy |
| aablocks | AA001K69 | AZD3965 98% | 25mg | $170 | 2026-05-28 | Buy |
| aablocks | AA001K69 | AZD3965 95% | 250mg | $1130 | 2026-05-28 | Buy |
| ACHEMBLOCK | M22559 | AZD3965 98% | 1G | $2450 | 2026-05-27 | Buy |
| ACHEMBLOCK | M22559 | AZD3965 98% | 25MG | $180 | 2026-05-27 | Buy |
| ACHEMBLOCK | M22559 | AZD3965 98% | 5MG | $65 | 2026-05-27 | Buy |
| ACHEMBLOCK | M22559 | AZD3965 98% | 100MG | $495 | 2026-05-27 | Buy |
| AK Scientific | 7027CR | CID10369242 | 50mg | $758 | 2021-12-16 | Buy |
| ApexBio Technology | C5049 | AZD 3965 | 10mg | $240 | 2026-05-06 | Buy |
| ApexBio Technology | C5049 | AZD 3965 | 25mg | $430 | 2026-05-06 | Buy |
| ApexBio Technology | C5049 | AZD 3965 | 5mg | $150 | 2026-05-06 | Buy |
| Arctom | HY-12750 | AZD3965 99.93% | 10mM*1mLinDMSO(Solution) | $155 | 2026-05-26 | Buy |
| Arctom | HY-12750 | AZD3965 99.93% | 10mg | $171 | 2026-05-26 | Buy |
Properties
Boiling point :723.1±70.0 °C(Predicted)
Density :1.483±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :insoluble in H2O; ≥51.5 mg/mL in DMSO; ≥51.6 mg/mL in EtOH
form :A crystalline solid
pka :10.92±0.50(Predicted)
color :White to off-white
InChIKey :PRNXOFBDXNTIFG-FQEVSTJZSA-N
SMILES :C1(=O)N(C)C(=O)C2C(C(N3C[C@@](O)(C)CO3)=O)=C(CC3=C(C)NN=C3C(F)(F)F)SC=2N1C(C)C
Density :1.483±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :insoluble in H2O; ≥51.5 mg/mL in DMSO; ≥51.6 mg/mL in EtOH
form :A crystalline solid
pka :10.92±0.50(Predicted)
color :White to off-white
InChIKey :PRNXOFBDXNTIFG-FQEVSTJZSA-N
SMILES :C1(=O)N(C)C(=O)C2C(C(N3C[C@@](O)(C)CO3)=O)=C(CC3=C(C)NN=C3C(F)(F)F)SC=2N1C(C)C
Safety Information
| Symbol(GHS): |
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| Signal word: | Warning | ||||||||||||||
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Description
AZD 3965 is a potent inhibitor of monocarboxylate transporter 1 (MCT1; Ki = 1.6 nM), killing tumor cells that are reliant on glycolysis by blocking lactate transport. It displays six-fold selectivity for MCT1 over MCT2 and is without effect against MCT4 at 10 μM. AZD 3965 increases intratumor lactate levels and decreases tumor growth in mice bearing COR-L103 small cell lung cancer (SCLC) xenografts. AZD 3965 also enhances radiosensitivity in mice with SCLC xenografts.More related product prices
(S)-6-[(3,5-Dimethyl-1H-pyrazol-4-yl)methyl]-5-[(4-hydroxyisoxazolidin-2-yl)carbonyl]-1-isobutyl-3-methylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione AZD3965 1-(4-(5-(5-amino-6-(5-(tert-butyl)-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-oneRelated product price
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(S)-6-[(3,5-Dimethyl-1H-pyrazol-4-yl)methyl]-5-[(4-hydroxyisoxazolidin-2-yl)carbonyl]-1-isobutyl-3-methylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione
$51-11227.7 -
AZD3965
$27-5672 -
1-(4-(5-(5-amino-6-(5-(tert-butyl)-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one
$41-2600
Suppliers and manufacturers
BOC Sciences
Zhejiang J&C Biological Technology Co.,Limited
TargetMol Chemicals Inc.
Zibo Hangyu Biotechnology Development Co., Ltd
HANGZHOU LEAP CHEM CO., LTD.
Aladdin Scientific
Amadis Chemical Company Limited
Chembest Research Laboratories Limited
Nanjing Chemlin Chemical Co., Ltd
![5-{[(4S)-4-Hydroxy-4-methyl-1,2-oxazolidin-2-yl]carbonyl}-1-isopropyl-3-methyl-6-{[5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]methyl}thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione](https://img.chemicalbook.com/ProductImageEN/2020-1/small/d18f9122-cb5f-4c28-b842-cfdc5c88dfe7.png){kind=small}