Astemizole
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- $39 - $1015
- Product name: Astemizole
- CAS: 68844-77-9
- MF: C28H31FN4O
- MW: 458.57
- EINECS:272-441-9
- MDL Number:MFCD00153919
- Synonyms:1-((4-fluorophenyl)methyl)-n-(1-(2-(4-methoxyphenyl)ethyl)-4-piperidinyl)-1h-b ;r45312 ;retolen ;ASTEMIZOLE;1-[(4-FLUOROPHENYL)METHYL]-N-[1-[2-(4-METHOXYPHENYL)ETHYL]-4-PIPERIDINYL]-1H-BENZIMIDAZOL-2-AMINE;(1-[4-FLUOROBENZYL]-2-[1-(4-METHOXYPHENETHYL)PIPERIDIN-4-YL] AMINOBENZIMIDAZOLE;Astemisan;R 43512
26 prices
Selected condition：
Brand
- AK Scientific
- Alfa Aesar
- American Custom Chemicals Corporation
- ApexBio Technology
- AvaChem
- Biosynth Carbosynth
- Cayman Chemical
- ChemScene
- DC Chemicals
- Medical Isotopes, Inc.
- Oakwood
- Sigma-Aldrich
- Tocris
- TRC
Package
- 50
- 5mg
- 10mg
- 25MG
- 50mg
- 100mg
- 250mg
- 1g
- ManufacturerAK Scientific
- Product numberK146
- Product descriptionAstemizole
- Packaging10mg
- Price$104
- Updated2021-12-16
- Buy
- ManufacturerAlfa Aesar
- Product numberJ60339
- Product descriptionAstemizole, 99+%
- Packaging50mg
- Price$171.65
- Updated2024-03-01
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0002918
- Product descriptionASTEMIZOLE 95.00%
- Packaging10MG
- Price$165.9
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0002918
- Product descriptionASTEMIZOLE 95.00%
- Packaging25MG
- Price$704.55
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB7409
- Product descriptionAstemizole
- Packaging100mg
- Price$140
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number3753
- Product descriptionAstemizole
- Packaging10mg
- Price$39
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number3753
- Product descriptionAstemizole
- Packaging25mg
- Price$59
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number3753
- Product descriptionAstemizole
- Packaging100mg
- Price$139
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFA18002
- Product descriptionAstemizole
- Packaging10mg
- Price$41
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFA18002
- Product descriptionAstemizole
- Packaging25mg
- Price$75
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFA18002
- Product descriptionAstemizole
- Packaging50mg
- Price$99
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number16967
- Product descriptionAstemizole ≥98%
- Packaging25mg
- Price$49
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16967
- Product descriptionAstemizole ≥98%
- Packaging50mg
- Price$92
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16967
- Product descriptionAstemizole ≥98%
- Packaging100mg
- Price$172
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-0011989
- Product descriptionAstemizole 99.68%
- Packaging5mg
- Price$50
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-0011989
- Product descriptionAstemizole 99.68%
- Packaging10mg
- Price$70
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | K146 | Astemizole | 10mg | $104 | 2021-12-16 | Buy |
| Alfa Aesar | J60339 | Astemizole, 99+% | 50mg | $171.65 | 2024-03-01 | Buy |
| American Custom Chemicals Corporation | API0002918 | ASTEMIZOLE 95.00% | 10MG | $165.9 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0002918 | ASTEMIZOLE 95.00% | 25MG | $704.55 | 2021-12-16 | Buy |
| ApexBio Technology | B7409 | Astemizole | 100mg | $140 | 2021-12-16 | Buy |
| AvaChem | 3753 | Astemizole | 10mg | $39 | 2021-12-16 | Buy |
| AvaChem | 3753 | Astemizole | 25mg | $59 | 2021-12-16 | Buy |
| AvaChem | 3753 | Astemizole | 100mg | $139 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FA18002 | Astemizole | 10mg | $41 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FA18002 | Astemizole | 25mg | $75 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FA18002 | Astemizole | 50mg | $99 | 2021-12-16 | Buy |
| Cayman Chemical | 16967 | Astemizole ≥98% | 25mg | $49 | 2024-03-01 | Buy |
| Cayman Chemical | 16967 | Astemizole ≥98% | 50mg | $92 | 2024-03-01 | Buy |
| Cayman Chemical | 16967 | Astemizole ≥98% | 100mg | $172 | 2024-03-01 | Buy |
| ChemScene | CS-0011989 | Astemizole 99.68% | 5mg | $50 | 2021-12-16 | Buy |
| ChemScene | CS-0011989 | Astemizole 99.68% | 10mg | $70 | 2021-12-16 | Buy |
Properties
Melting point :172.9°C
Boiling point :627.3±65.0 °C(Predicted)
Density :1.1587 (estimate)
storage temp. :2-8°C
solubility :DMSO: >20mg/mL
pka :pKa 4.85(H2O t=25.0 I=0.025) (Uncertain);8.69(H2O t=25.0 I=0.025) (Uncertain)
form :powder
color :Crystals
Water Solubility :It is soluble in DMSO (25 mg/ml ), ethanol (25 mg/ml), chloroform, methanol, and water (partly miscible).
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
Boiling point :627.3±65.0 °C(Predicted)
Density :1.1587 (estimate)
storage temp. :2-8°C
solubility :DMSO: >20mg/mL
pka :pKa 4.85(H2O t=25.0 I=0.025) (Uncertain);8.69(H2O t=25.0 I=0.025) (Uncertain)
form :powder
color :Crystals
Water Solubility :It is soluble in DMSO (25 mg/ml ), ethanol (25 mg/ml), chloroform, methanol, and water (partly miscible).
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
Safety Information
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Description
Astemizole is a non-sedating antihistamine that antagonizes the histamine H1 receptor with a Ki value of 4.4 nM. It is considerably less potent at muscarinic acetylcholine receptors (Ki = 2.4 μM). Astemizole is also a potent blocker of ether-a-go-go-related gene (ERG) potassium channels (IC50 = ~1 nM) that has been used to study long QT syndrome type 2. Furthermore, because it can target oncogenic ERG1 and ERG potassium channels, astemizole has been explored as a potential antineoplastic agent for decreasing proliferation of various cancer cells.More related product prices
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Suppliers and manufacturers
Henan Tianfu Chemical Co.,Ltd.
ATK CHEMICAL COMPANY LIMITED
CONIER CHEM AND PHARMA LIMITED
TargetMol Chemicals Inc.
Shaanxi Dideu Medichem Co. Ltd
AFINE CHEMICALS LIMITED
Zhejiang J&C Biological Technology Co.,Limited
