BAZEDOXIFENE ACETATE
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- $39 - $2691.1
- Product name: BAZEDOXIFENE ACETATE
- CAS: 198481-33-3
- MF: C32H38N2O5
- MW: 530.67
- EINECS:638-804-4
- MDL Number:MFCD09260074
- Synonyms:BAZEDOXIFENE ACETATE;1-(p-(2-(Hexahydro-1H-azepin-1-yl)ethoxy)benzyl)-2-(p-hydroxyphenyl)-3-methylindol-5-ol monoacetate (salt);1H-Indol-5-ol, 1-((4-(2-(hexahydro-1H-azepin-1-yl)ethoxy)phenyl)methyl)-2-(4-hydroxyphenyl)-3-methyl-, monoacetate (salt);Bazedoxifene acetate [usan];Unii-J70472ud3d;Viviant;Way-140424;1-((4-(2-(Hexahydro-1H-azepin-1-yl)ethoxy)phenyl)methyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-ol monoacetate
34 prices
Selected condition：
Brand
- AK Scientific
- Ambeed
- ApexBio Technology
- Biorbyt Ltd
- Biosynth Carbosynth
- Cayman Chemical
- Chemcia Scientific
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Medical Isotopes, Inc.
- Sigma-Aldrich
- Tocris
- TRC
Package
- 50
- 5mg
- 1mg
- 10
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 0.5g
- 1g
- 1000mg
- ManufacturerAK Scientific
- Product numberY0396
- Product descriptionBazedoxifene acetate
- Packaging5mg
- Price$39
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA688355
- Product description1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99%
- Packaging10mg
- Price$40
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA688355
- Product description1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99%
- Packaging50mg
- Price$66
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA688355
- Product description1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99%
- Packaging100mg
- Price$85
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA688355
- Product description1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99%
- Packaging250mg
- Price$130
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA688355
- Product description1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99%
- Packaging1g
- Price$316
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA3233
- Product descriptionBazedoxifene acetate
- Packaging10mg
- Price$140
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181209
- Product descriptionBazedoxifene acetate >98%
- Packaging100mg
- Price$690.2
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181209
- Product descriptionBazedoxifene acetate >98%
- Packaging250mg
- Price$1356.6
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181209
- Product descriptionBazedoxifene acetate >98%
- Packaging1000mg
- Price$2691.1
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFB45398
- Product descriptionBazedoxifene acetate
- Packaging100mg
- Price$125
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFB45398
- Product descriptionBazedoxifene acetate
- Packaging250mg
- Price$200
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number15005
- Product descriptionBazedoxifene acetate ≥98%
- Packaging5mg
- Price$111
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15005
- Product descriptionBazedoxifene acetate ≥98%
- Packaging10mg
- Price$210
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15005
- Product descriptionBazedoxifene acetate ≥98%
- Packaging25mg
- Price$493
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number15005
- Product descriptionBazedoxifene acetate ≥98%
- Packaging50mg
- Price$765
- Updated2024-03-01
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | Y0396 | Bazedoxifene acetate | 5mg | $39 | 2021-12-16 | Buy |
| Ambeed | A688355 | 1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99% | 10mg | $40 | 2021-12-16 | Buy |
| Ambeed | A688355 | 1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99% | 50mg | $66 | 2021-12-16 | Buy |
| Ambeed | A688355 | 1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99% | 100mg | $85 | 2021-12-16 | Buy |
| Ambeed | A688355 | 1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99% | 250mg | $130 | 2021-12-16 | Buy |
| Ambeed | A688355 | 1-(4-(2-(Azepan-1-yl)ethoxy)benzyl)-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-olacetate 99% | 1g | $316 | 2021-12-16 | Buy |
| ApexBio Technology | A3233 | Bazedoxifene acetate | 10mg | $140 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181209 | Bazedoxifene acetate >98% | 100mg | $690.2 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181209 | Bazedoxifene acetate >98% | 250mg | $1356.6 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181209 | Bazedoxifene acetate >98% | 1000mg | $2691.1 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FB45398 | Bazedoxifene acetate | 100mg | $125 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FB45398 | Bazedoxifene acetate | 250mg | $200 | 2021-12-16 | Buy |
| Cayman Chemical | 15005 | Bazedoxifene acetate ≥98% | 5mg | $111 | 2024-03-01 | Buy |
| Cayman Chemical | 15005 | Bazedoxifene acetate ≥98% | 10mg | $210 | 2024-03-01 | Buy |
| Cayman Chemical | 15005 | Bazedoxifene acetate ≥98% | 25mg | $493 | 2024-03-01 | Buy |
| Cayman Chemical | 15005 | Bazedoxifene acetate ≥98% | 50mg | $765 | 2024-03-01 | Buy |
Properties
Melting point :174-178°
storage temp. :-20°C
solubility :DMSO: soluble15mg/mL, clear
form :powder
color :white to beige
InChIKey :DGEPGJZKMFNSDD-UHFFFAOYSA-N
SMILES :C(=O)(O)C.C(C1C=CC(OCCN2CCCCCC2)=CC=1)N1C2C=CC(O)=CC=2C(C)=C1C1C=CC(O)=CC=1
storage temp. :-20°C
solubility :DMSO: soluble15mg/mL, clear
form :powder
color :white to beige
InChIKey :DGEPGJZKMFNSDD-UHFFFAOYSA-N
SMILES :C(=O)(O)C.C(C1C=CC(OCCN2CCCCCC2)=CC=1)N1C2C=CC(O)=CC=2C(C)=C1C1C=CC(O)=CC=1
Safety Information
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| Signal word: | Warning | ||||||||||||||||||||||||||||
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Description
Bazedoxifene acetate is a third generation selective estrogen receptor modulator (SERM). It is an indole-based ER ligand that binds to both ERα (IC50 = 26 nM) and ERβ (IC50 = 99 nM). Bazedoxifene actetate antagonizes 17β-estradiol-dependent MCF-7 and T47D breast cancer cell proliferation in vitro as well as hormone-independent growth of MCF-7:5C cells that are resistant to long-term estrogen deprivation (80% reduction with 10 nM). It has been shown to arrest cell cycling by downregulating cyclin D1 and ERα.More related product prices
4-[2-(1-AZEPANYL)ETHOXY]BENZYL CHLORIDE HCL BenzeneMethanol, 4-[2-(hexahydro-1H-azepin-1-yl)ethoxy]- (hydrochloride) 3-METHYL-5-(PHENYLMETHOXY)-2-[4-(PHENYLMETHOXY)PHENYL]-1H-INDOLE 1-[4-(2-AZEPAN-1-YL-ETHOXY)-BENZYL]-5-BENZYLOXY-2-(4-BENZYLOXY-PHENYL)-3-METHYL-1H-INDOLE Tolvaptan Bazedoxifene 4’-β-D-Glucuronide Hyaluronic acid Sodium tripolyphosphate Sodium metaphosphate 1-[[4-[2-(Hexahydro-1H-azepin-1-yl)(ethoxy-d4)]phenyl]Methyl]-2-(4-hydroxyphenyl)-3-Methyl-