BQ-788
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- $76 - $6200
- Product name: BQ-788
- CAS: 156161-89-6
- MF: C34H52N5NaO7
- MW: 665.81
- EINECS:
- MDL Number:MFCD00797882
- Synonyms:BQ-788 SODIUM;BQ-788 SYNTHETIC >97% ETB ENDOTHELIN REC EPT;N-[(cis-2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucinesodiumsalt;1-ELAIDYLPHOSPHOCHOLINE, >97%;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl]-1-(methoxycarbonyl)-D-tryptophyl]-D-norleucine sodium salt, 2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-;DMpc-gaMMa-MeLeu-D-Trp(1-CO2CH3)-D-Nle.Na (DMpc : cis-2,6-DiMethylpiperidinocarbonyl);2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
50 prices
Selected condition:
Brand
- aablocks
- Adipogen Life Sciences
- AK Scientific
- Alichem
- ApexBio Technology
- Arctom
- AvaChem
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Sigma-Aldrich
- TRC
- Usbiological
Package
- 1mg
- 50mg
- 100mg
- 250mg
- 1g
- 10mM(in1mLDMSO)
- 200μg
- 500μg
- 5mg
- 10mg
- 25mg
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging1mg
- Price$76
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging5mg
- Price$174
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging10mg
- Price$250
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging25mg
- Price$500
- Updated2026-05-28
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CP3-0012-M001
- Product descriptionBQ-788 . sodium salt ≥95%(HPLC)
- Packaging1mg
- Price$220
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CP3-0012-M001
- Product descriptionBQ-788.sodiumsalt ≥95%(HPLC)
- Packaging1mg
- Price$200
- Updated2021-12-16
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CP3-0012-C500
- Product descriptionBQ-788 . sodium salt ≥95%(HPLC)
- Packaging500μg
- Price$150
- Updated2026-05-06
- Buy
- ManufacturerAK Scientific
- Product number3506AH
- Product descriptionDMPC-Gamma-MELEU-D-Trp(1-Co2CH3)-D-NleNa
- Packaging1mg
- Price$368
- Updated2021-12-16
- Buy
- ManufacturerAlichem
- Product number156161896
- Product descriptionSodiumBQ-788
- Packaging10mg
- Price$400
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging10mM(in1mLDMSO)
- Price$392
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging5mg
- Price$327
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging10mg
- Price$450
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging1mg
- Price$148
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberHY-15894
- Product descriptionBQ-788sodiumsalt 99.33%
- Packaging1mg
- Price$124
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15894
- Product descriptionBQ-788sodiumsalt 99.33%
- Packaging5mg
- Price$285
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15894
- Product descriptionBQ-788sodiumsalt 99.33%
- Packaging25mg
- Price$817
- Updated2026-05-26
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 1mg | $76 | 2026-05-28 | Buy |
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 5mg | $174 | 2026-05-28 | Buy |
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 10mg | $250 | 2026-05-28 | Buy |
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 25mg | $500 | 2026-05-28 | Buy |
| Adipogen Life Sciences | AG-CP3-0012-M001 | BQ-788 . sodium salt ≥95%(HPLC) | 1mg | $220 | 2026-05-06 | Buy |
| Adipogen Life Sciences | AG-CP3-0012-M001 | BQ-788.sodiumsalt ≥95%(HPLC) | 1mg | $200 | 2021-12-16 | Buy |
| Adipogen Life Sciences | AG-CP3-0012-C500 | BQ-788 . sodium salt ≥95%(HPLC) | 500μg | $150 | 2026-05-06 | Buy |
| AK Scientific | 3506AH | DMPC-Gamma-MELEU-D-Trp(1-Co2CH3)-D-NleNa | 1mg | $368 | 2021-12-16 | Buy |
| Alichem | 156161896 | SodiumBQ-788 | 10mg | $400 | 2021-12-16 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 10mM(in1mLDMSO) | $392 | 2026-05-06 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 5mg | $327 | 2026-05-06 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 10mg | $450 | 2026-05-06 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 1mg | $148 | 2026-05-06 | Buy |
| Arctom | HY-15894 | BQ-788sodiumsalt 99.33% | 1mg | $124 | 2026-05-26 | Buy |
| Arctom | HY-15894 | BQ-788sodiumsalt 99.33% | 5mg | $285 | 2026-05-26 | Buy |
| Arctom | HY-15894 | BQ-788sodiumsalt 99.33% | 25mg | $817 | 2026-05-26 | Buy |
Properties
storage temp. :-20°C
solubility :acetonitrile: 0.3 mg/mL
form :solid
color :white
Water Solubility :acetonitrile: 0.3mg/mL
DMSO: 1.2mg/mL
ethanol: 1.2mg/mL
H2O: slightly soluble InChIKey :IBWYJVKAVOHKHB-IAZAOAQXNA-N
SMILES :C(C1=CN(C(=O)OC)C2=CC=CC=C12)[C@H](C(=O)N[C@@H](C(=O)O)CCCC)NC(=O)[C@H](CC(C)(C)C)NC(N1[C@@H](CCC[C@@H]1C)C)=O.[NaH] |&1:14,18,29,38,42,r|
solubility :acetonitrile: 0.3 mg/mL
form :solid
color :white
Water Solubility :acetonitrile: 0.3mg/mL
DMSO: 1.2mg/mL
ethanol: 1.2mg/mL
H2O: slightly soluble InChIKey :IBWYJVKAVOHKHB-IAZAOAQXNA-N
SMILES :C(C1=CN(C(=O)OC)C2=CC=CC=C12)[C@H](C(=O)N[C@@H](C(=O)O)CCCC)NC(=O)[C@H](CC(C)(C)C)NC(N1[C@@H](CCC[C@@H]1C)C)=O.[NaH] |&1:14,18,29,38,42,r|
Safety Information
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Description
The endothelin (ET) family of proteins mediate a variety of responses, with ET-1 being a potent and long-lasting constrictor of human cardiovascular vessels. These proteins activate the G protein-coupled receptors ETA and ETB, with ETB being non-specific for ET protein form. BQ-788 is a potent, selective antagonist of ETB (IC50 = 1.2 nM for blocking ET-1 binding to human Girardi heart cells). It weakly inhibits the binding of ET-1 to ETA receptors on human neuroblastoma SK-N-MC cells (IC50 = 1300 nM). BQ-788 competitively antagonizes the vasoconstriction induced by an ETB-selective agonist on isolated rabbit pulmonary arteries, blocks ET-1 induced bronchoconstriction in guinea pigs, and abolishes an ET-1 mediated depressor response in rats.Related product price
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