BQ-788
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- $76 - $6200
- Product name: BQ-788
- CAS: 156161-89-6
- MF: C34H52N5NaO7
- MW: 665.81
- EINECS:
- MDL Number:MFCD00797882
- Synonyms:BQ-788 SODIUM;BQ-788 SYNTHETIC >97% ETB ENDOTHELIN REC EPT;N-[(cis-2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucinesodiumsalt;1-ELAIDYLPHOSPHOCHOLINE, >97%;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl]-1-(methoxycarbonyl)-D-tryptophyl]-D-norleucine sodium salt, 2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle;N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-;DMpc-gaMMa-MeLeu-D-Trp(1-CO2CH3)-D-Nle.Na (DMpc : cis-2,6-DiMethylpiperidinocarbonyl);2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
40 prices
Selected condition:
Brand
- aablocks
- Adipogen Life Sciences
- AK Scientific
- Alichem
- ApexBio Technology
- Arctom
- AvaChem
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Sigma-Aldrich
- TRC
- Usbiological
Package
- 5mg
- 50mg
- 100mg
- 250mg
- 1g
- 10mM(in1mLDMSO)
- 200μg
- 500μg
- 1mg
- 10mg
- 25mg
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging5mg
- Price$174
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging10mg
- Price$250
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging25mg
- Price$500
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001OHP
- Product descriptionSodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98%
- Packaging1mg
- Price$76
- Updated2026-05-28
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CP3-0012-M001
- Product descriptionBQ-788 . sodium salt ≥95%(HPLC)
- Packaging1mg
- Price$220
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CP3-0012-C500
- Product descriptionBQ-788 . sodium salt ≥95%(HPLC)
- Packaging500μg
- Price$150
- Updated2026-05-06
- Buy
- ManufacturerAK Scientific
- Product number3506AH
- Product descriptionDMPC-Gamma-MELEU-D-Trp(1-Co2CH3)-D-NleNa
- Packaging1mg
- Price$368
- Updated2021-12-16
- Buy
- ManufacturerAlichem
- Product number156161896
- Product descriptionSodiumBQ-788
- Packaging10mg
- Price$400
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging10mM(in1mLDMSO)
- Price$392
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging10mg
- Price$450
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging1mg
- Price$148
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB3278
- Product descriptionBQ-788 sodium salt
- Packaging5mg
- Price$327
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberHY-15894
- Product descriptionBQ-788sodiumsalt 99.33%
- Packaging5mg
- Price$285
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15894
- Product descriptionBQ-788sodiumsalt 99.33%
- Packaging1mg
- Price$124
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15894
- Product descriptionBQ-788sodiumsalt 99.33%
- Packaging10mg
- Price$409
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15894
- Product descriptionBQ-788sodiumsalt 99.33%
- Packaging50mg
- Price$1308
- Updated2026-05-26
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 5mg | $174 | 2026-05-28 | Buy |
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 10mg | $250 | 2026-05-28 | Buy |
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 25mg | $500 | 2026-05-28 | Buy |
| aablocks | AA001OHP | Sodium N-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucine 98% | 1mg | $76 | 2026-05-28 | Buy |
| Adipogen Life Sciences | AG-CP3-0012-M001 | BQ-788 . sodium salt ≥95%(HPLC) | 1mg | $220 | 2026-05-06 | Buy |
| Adipogen Life Sciences | AG-CP3-0012-C500 | BQ-788 . sodium salt ≥95%(HPLC) | 500μg | $150 | 2026-05-06 | Buy |
| AK Scientific | 3506AH | DMPC-Gamma-MELEU-D-Trp(1-Co2CH3)-D-NleNa | 1mg | $368 | 2021-12-16 | Buy |
| Alichem | 156161896 | SodiumBQ-788 | 10mg | $400 | 2021-12-16 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 10mM(in1mLDMSO) | $392 | 2026-05-06 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 10mg | $450 | 2026-05-06 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 1mg | $148 | 2026-05-06 | Buy |
| ApexBio Technology | B3278 | BQ-788 sodium salt | 5mg | $327 | 2026-05-06 | Buy |
| Arctom | HY-15894 | BQ-788sodiumsalt 99.33% | 5mg | $285 | 2026-05-26 | Buy |
| Arctom | HY-15894 | BQ-788sodiumsalt 99.33% | 1mg | $124 | 2026-05-26 | Buy |
| Arctom | HY-15894 | BQ-788sodiumsalt 99.33% | 10mg | $409 | 2026-05-26 | Buy |
| Arctom | HY-15894 | BQ-788sodiumsalt 99.33% | 50mg | $1308 | 2026-05-26 | Buy |
Properties
storage temp. :-20°C
solubility :acetonitrile: 0.3 mg/mL
form :solid
color :white
Water Solubility :acetonitrile: 0.3mg/mL
DMSO: 1.2mg/mL
ethanol: 1.2mg/mL
H2O: slightly soluble InChIKey :IBWYJVKAVOHKHB-IAZAOAQXNA-N
SMILES :C(C1=CN(C(=O)OC)C2=CC=CC=C12)[C@H](C(=O)N[C@@H](C(=O)O)CCCC)NC(=O)[C@H](CC(C)(C)C)NC(N1[C@@H](CCC[C@@H]1C)C)=O.[NaH] |&1:14,18,29,38,42,r|
solubility :acetonitrile: 0.3 mg/mL
form :solid
color :white
Water Solubility :acetonitrile: 0.3mg/mL
DMSO: 1.2mg/mL
ethanol: 1.2mg/mL
H2O: slightly soluble InChIKey :IBWYJVKAVOHKHB-IAZAOAQXNA-N
SMILES :C(C1=CN(C(=O)OC)C2=CC=CC=C12)[C@H](C(=O)N[C@@H](C(=O)O)CCCC)NC(=O)[C@H](CC(C)(C)C)NC(N1[C@@H](CCC[C@@H]1C)C)=O.[NaH] |&1:14,18,29,38,42,r|
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||||||||||||||||
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Description
The endothelin (ET) family of proteins mediate a variety of responses, with ET-1 being a potent and long-lasting constrictor of human cardiovascular vessels. These proteins activate the G protein-coupled receptors ETA and ETB, with ETB being non-specific for ET protein form. BQ-788 is a potent, selective antagonist of ETB (IC50 = 1.2 nM for blocking ET-1 binding to human Girardi heart cells). It weakly inhibits the binding of ET-1 to ETA receptors on human neuroblastoma SK-N-MC cells (IC50 = 1300 nM). BQ-788 competitively antagonizes the vasoconstriction induced by an ETB-selective agonist on isolated rabbit pulmonary arteries, blocks ET-1 induced bronchoconstriction in guinea pigs, and abolishes an ET-1 mediated depressor response in rats.Related product price
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BQ-788
$76-6200 -
4277-63-8
$19-1397 -
AC-D-NLE-OH
$33-1247
Suppliers and manufacturers
Hangzhou Sinoda Pharmaceutical Technology Co. LTD
3B Pharmachem (Wuhan) International Co.,Ltd.
Shanghai Sinch Parmaceuticals Tech. Co. Ltd.
Chemsky(shanghai)International Co.,Ltd.
Haoyuan Chemexpress Co., Ltd.
AdooQ BioScience, LLC
ShangHai Caerulum Pharma Discovery Co., Ltd.
Bide Pharmatech Ltd.
AdooQ Bioscience CHINA
Sigma-Aldrich




