GSK 2801
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- $32 - $1677
- Product name: GSK 2801
- CAS: 1619994-68-1
- MF: C20H21NO4S
- MW: 371.45
- EINECS:
- MDL Number:MFCD26142953
- Synonyms:GSK 2801;GSK2801;GSK-2801;1-(7-(2-Methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone;1-(1-(2-(methylsulfonyl)phenyl)-7-propoxyindolizin-3-yl)ethanone;1-[1-[2-(Methylsulfonyl)phenyl]-7-propoxy-3-indolizinyl]ethanone;Ethanone, 1-[1-[2-(methylsulfonyl)phenyl]-7-propoxy-3-indolizinyl]-;GSK-2801; GSK 280
39 prices
Selected condition：
Brand
- ACHEMBLOCK
- AK Scientific
- ApexBio Technology
- Arctom
- Biosynth
- BroadPharm
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Sigma-Aldrich
- Tocris
- TRC
- Usbiological
Package
- 1mg
- 10mg
- 25mg
- 10mM*1mLinDMSO(Solid+Solvent)
- 10
- 5mg
- 50mg
- 10mM*1mLinDMSO
- 250mg
- 1g
- 5 mg
- 25 mg
- 10mM*1mLinDMSO(Solution)
- 100MG
- 10mM(in 1mL DMSO)
- 10mM(in1mLDMSO)
- ManufacturerACHEMBLOCK
- Product numberO33849
- Product descriptionGSK2801 98%
- Packaging100MG
- Price$160
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product number3707AH
- Product description1-(7-(2-Methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone
- Packaging1g
- Price$1185
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB5998
- Product descriptionGSK2801
- Packaging50mg
- Price$305
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB5998
- Product descriptionGSK2801
- Packaging50mg
- Price$336
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB5998
- Product descriptionGSK2801
- Packaging10mM(in 1mL DMSO)
- Price$50
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB5998
- Product descriptionGSK2801
- Packaging10mg
- Price$75
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB5998
- Product descriptionGSK2801
- Packaging10mg
- Price$83
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB5998
- Product descriptionGSK2801
- Packaging10mM(in1mLDMSO)
- Price$88
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberHY-15658
- Product descriptionGSK2801 99.69%
- Packaging10mM*1mLinDMSO(Solution)
- Price$92
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15658
- Product descriptionGSK2801 99.69%
- Packaging10mg
- Price$115
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15658
- Product descriptionGSK2801 99.69%
- Packaging5mg
- Price$84
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15658
- Product descriptionGSK2801 99.69%
- Packaging10mM*1mLinDMSO(Solid+Solvent)
- Price$87
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15658
- Product descriptionGSK2801 99.69%
- Packaging25mg
- Price$262
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15658
- Product descriptionGSK2801 99.69%
- Packaging50mg
- Price$418
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-15658
- Product descriptionGSK2801 99.69%
- Packaging100mg
- Price$627
- Updated2026-05-26
- Buy
- ManufacturerBiosynth
- Product numberFG137682
- Product descriptionGSK 2801
- Packaging50mg
- Price$437.5
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| ACHEMBLOCK | O33849 | GSK2801 98% | 100MG | $160 | 2026-05-27 | Buy |
| AK Scientific | 3707AH | 1-(7-(2-Methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone | 1g | $1185 | 2021-12-16 | Buy |
| ApexBio Technology | B5998 | GSK2801 | 50mg | $305 | 2021-12-16 | Buy |
| ApexBio Technology | B5998 | GSK2801 | 50mg | $336 | 2026-05-06 | Buy |
| ApexBio Technology | B5998 | GSK2801 | 10mM(in 1mL DMSO) | $50 | 2021-12-16 | Buy |
| ApexBio Technology | B5998 | GSK2801 | 10mg | $75 | 2021-12-16 | Buy |
| ApexBio Technology | B5998 | GSK2801 | 10mg | $83 | 2026-05-06 | Buy |
| ApexBio Technology | B5998 | GSK2801 | 10mM(in1mLDMSO) | $88 | 2026-05-06 | Buy |
| Arctom | HY-15658 | GSK2801 99.69% | 10mM*1mLinDMSO(Solution) | $92 | 2026-05-26 | Buy |
| Arctom | HY-15658 | GSK2801 99.69% | 10mg | $115 | 2026-05-26 | Buy |
| Arctom | HY-15658 | GSK2801 99.69% | 5mg | $84 | 2026-05-26 | Buy |
| Arctom | HY-15658 | GSK2801 99.69% | 10mM*1mLinDMSO(Solid+Solvent) | $87 | 2026-05-26 | Buy |
| Arctom | HY-15658 | GSK2801 99.69% | 25mg | $262 | 2026-05-26 | Buy |
| Arctom | HY-15658 | GSK2801 99.69% | 50mg | $418 | 2026-05-26 | Buy |
| Arctom | HY-15658 | GSK2801 99.69% | 100mg | $627 | 2026-05-26 | Buy |
| Biosynth | FG137682 | GSK 2801 | 50mg | $437.5 | 2021-12-16 | Buy |
Properties
Density :1.23±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :insoluble in H2O; ≥18.55 mg/mL in DMSO; ≥2.82 mg/mL in EtOH with gentle warming and ultrasonic
form :solid
color :Light yellow to khaki
InChI :1S/C20H21NO4S/c1-4-11-25-15-9-10-21-18(14(2)22)13-17(19(21)12-15)16-7-5-6-8-20(16)26(3,23)24/h5-10,12-13H,4,11H2,1-3H3
InChIKey :KHWCPNJRJCNVRI-UHFFFAOYSA-N
SMILES :CCCOC1=CC2=C(C3=CC=CC=C3S(=O)(C)=O)C=C(C(C)=O)N2C=C1
storage temp. :-20°C
solubility :insoluble in H2O; ≥18.55 mg/mL in DMSO; ≥2.82 mg/mL in EtOH with gentle warming and ultrasonic
form :solid
color :Light yellow to khaki
InChI :1S/C20H21NO4S/c1-4-11-25-15-9-10-21-18(14(2)22)13-17(19(21)12-15)16-7-5-6-8-20(16)26(3,23)24/h5-10,12-13H,4,11H2,1-3H3
InChIKey :KHWCPNJRJCNVRI-UHFFFAOYSA-N
SMILES :CCCOC1=CC2=C(C3=CC=CC=C3S(=O)(C)=O)C=C(C(C)=O)N2C=C1
Safety Information
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| Signal word: | Warning | ||||||||||||||
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Description
BAZ2A/B are bromodomain-containing proteins whose biological function is believed to function similarly to ACF1, the Drosophila BAZ2B ortholog. ACF complexes play roles in establishing regular nucleosome spacing during chromatin assembly and influencing different remodeling outcomes at target loci. BAZ2A and BAZ2B constitute the central scaffolding protein of the nucleolar remodeling complex (NoRC) that regulates the expression of noncoding RNAs. GSK2801 is a selective, cell-permeable inhibitor of the BAZ2 family of bromodomain-containing proteins (IC50s = 9-350 nM in a BAZ2B AlphaScreen). It binds to BAZ2A and BAZ2B with Kd values of 0.26 and 0.14 μM, respectively, and does not interact with the bromodomains of BRD4(BD1), CREBBP, TRIM24/TIF1α, PB1(BD5), PCAF, or ATAD2. See the Structural Genomics Consortium (SGC) website for more information.Related product price
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Suppliers and manufacturers
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Wuhan Jingkang en Biomedical Technology Co., Ltd
Amadis Chemical Company Limited
