KENPAULLONE
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- $23 - $1802
- Product name: KENPAULLONE
- CAS: 142273-20-9
- MF: C16H11BrN2O
- MW: 327.18
- EINECS:
- MDL Number:MFCD02683595
- Synonyms:9-Bromo-7,12-dihydro-indolo[3,2-d][1]benzazepin-6(5H)-one, NSC 664704;9-BroMopaullone;9-BROMO-7,12-DIHYDRO-INDOLO[3,2-D][1]BENZAZEPIN-6(5H)-ONE;8-BROMO-7,12-DIHYDRO-INDOLO[3,2-D][1]-BENZAZEPIN-6(5H)-ONE;KENPAULLONE;NSC-664704;Kenpaullone 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one;9-bromo-7,12-dihydro-5H-indolo[3,2-d][1]benzazepin-6-one
104 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- Ambeed
- ApexBio Technology
- Arctom
- AvaChem
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TCI Chemical
- Tocris
- TRC
- Usbiological
Package
- 10mM*1mLinDMSO
- 10mM*1mLinDMSO(Solid+Solvent)
- 10mM*1mLinDMSO(Solution)
- 25mg
- 10
- 25.00mg
- 50.00mg
- 100.00mg
- 10mM(in 1mL DMSO)
- 1mg
- 5mg
- 10mg
- 50mg
- 10mM(in1mLDMSO)
- 100MG
- 250MG
- 1G
- Manufactureraablocks
- Product numberAA001I10
- Product description9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one ≥97%(HPLC)
- Packaging50mg
- Price$71
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001I10
- Product description9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one 98%
- Packaging10mg
- Price$35
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001I10
- Product description9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one 98%
- Packaging5mg
- Price$28
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001I10
- Product description9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one 98%
- Packaging1mg
- Price$23
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberQ65731
- Product description9-bromo-7,12-dihydrobenzo[2,3]azepino[4,5-b]indol-6(5H)-one 98%
- Packaging100MG
- Price$115
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberQ65731
- Product description9-bromo-7,12-dihydrobenzo[2,3]azepino[4,5-b]indol-6(5H)-one 98%
- Packaging250MG
- Price$230
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberQ65731
- Product description9-bromo-7,12-dihydrobenzo[2,3]azepino[4,5-b]indol-6(5H)-one 98%
- Packaging1G
- Price$600
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberX5716
- Product descriptionKenpaullone
- Packaging50mg
- Price$197
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging100mg
- Price$164
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging250mg
- Price$245
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging50mg
- Price$102
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging10mg
- Price$60
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging1mg
- Price$27
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging5mg
- Price$46
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging1g
- Price$634
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6720
- Product descriptionKenpaullone
- Packaging50mg
- Price$473
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA001I10 | 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one ≥97%(HPLC) | 50mg | $71 | 2026-05-28 | Buy |
| aablocks | AA001I10 | 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one 98% | 10mg | $35 | 2026-05-28 | Buy |
| aablocks | AA001I10 | 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one 98% | 5mg | $28 | 2026-05-28 | Buy |
| aablocks | AA001I10 | 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one 98% | 1mg | $23 | 2026-05-28 | Buy |
| ACHEMBLOCK | Q65731 | 9-bromo-7,12-dihydrobenzo[2,3]azepino[4,5-b]indol-6(5H)-one 98% | 100MG | $115 | 2026-05-27 | Buy |
| ACHEMBLOCK | Q65731 | 9-bromo-7,12-dihydrobenzo[2,3]azepino[4,5-b]indol-6(5H)-one 98% | 250MG | $230 | 2026-05-27 | Buy |
| ACHEMBLOCK | Q65731 | 9-bromo-7,12-dihydrobenzo[2,3]azepino[4,5-b]indol-6(5H)-one 98% | 1G | $600 | 2026-05-27 | Buy |
| AK Scientific | X5716 | Kenpaullone | 50mg | $197 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 100mg | $164 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 250mg | $245 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 50mg | $102 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 10mg | $60 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 1mg | $27 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 5mg | $46 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 1g | $634 | 2021-12-16 | Buy |
| ApexBio Technology | B6720 | Kenpaullone | 50mg | $473 | 2026-05-06 | Buy |
Properties
Melting point :>300°C (dec.)
Boiling point :613.0±45.0 °C(Predicted)
Density :1.596±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 18 mg/mL, clear, yellow
pka :14.29±0.20(Predicted)
form :Yellow-brown solid
color :yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChI :1S/C16H11BrN2O/c17-9-5-6-14-11(7-9)12-8-15(20)18-13-4-2-1-3-10(13)16(12)19-14/h1-7,19H,8H2,(H,18,20)
InChIKey :QQUXFYAWXPMDOE-UHFFFAOYSA-N
SMILES :Brc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1
CAS DataBase Reference :142273-20-9(CAS DataBase Reference)
Boiling point :613.0±45.0 °C(Predicted)
Density :1.596±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 18 mg/mL, clear, yellow
pka :14.29±0.20(Predicted)
form :Yellow-brown solid
color :yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChI :1S/C16H11BrN2O/c17-9-5-6-14-11(7-9)12-8-15(20)18-13-4-2-1-3-10(13)16(12)19-14/h1-7,19H,8H2,(H,18,20)
InChIKey :QQUXFYAWXPMDOE-UHFFFAOYSA-N
SMILES :Brc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1
CAS DataBase Reference :142273-20-9(CAS DataBase Reference)
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
Kenpaullone is an ATP-competitive inhibitor of several CDKs (cyclin-dependent kinases) as well as GSK-3β (glycogen synthase kinase 3β). It has been shown to inhibit GSK-3 with an IC50 value of 0.23 μM and CDK1/cyclin B, CDK2/cyclin A, CDK5/p25, and lymphocyte kinase with IC50 values of 0.4, 0.68, 0.85, and 0.47 μM, respectively. Due to the compound’s activity, Kenpaullone is useful in the study of cell cycle regulators. Kenpaullone is an inhibitor of cyclin E, ERK 2 and p35.Related product price
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Suppliers and manufacturers
ATK CHEMICAL COMPANY LIMITED
BOC Sciences
CONIER CHEM AND PHARMA LIMITED
SHANGHAI T&W PHARMACEUTICAL CO., LTD.
Tianjin Xinshengjiahe Science & Technology Development Co,.Ltd
HANGZHOU CLAP TECHNOLOGY CO.,LTD
Zhejiang J&C Biological Technology Co.,Limited
InvivoChem
