LY2940680
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- $15 - $5541
- Product name: LY2940680
- CAS: 1258861-20-9
- MF: C26H24F4N6O
- MW: 512.5
- EINECS:
- MDL Number:MFCD21609264
- Synonyms:Taladegib (LY2940680);4-Fluoro-N-methyl-N-[1-[4-(1-methyl-1H-pyrazol-5-yl)-1-phthalazinyl]-4-piperidinyl]-2-(trifluoromethyl)benzamide LY 2940680;LY2940680;LY2940680 (Taladegib);Taladegib;Taladegib hydrochloride;4-Fluoro-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-2-(trifluo;4-Fluoro-N-methyl-N-[1-[4-(1-methyl-1H-pyrazol-5-yl)-1-phthalazinyl]-4-piperidinyl]-2-(trifluoromethyl)benzamide
71 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Axon Medchem
- Biorbyt Ltd
- Cayman Chemical
- Chemenu
- ChemScene
- Crysdot
- DC Chemicals
- Matrix Scientific
- TRC
Package
- 10mM*1mLinDMSO(Solid+Solvent)
- 2.5mg
- 10mM*1mLinDMSO(Solution)
- 1mg
- 10mM*1mLinDMSO
- 5mg
- 10mg
- 25MG
- 50mg
- 100MG
- 200mg
- 200.00mg
- 250mg
- 1000mg
- 1.00g
- 1G
- Manufactureraablocks
- Product numberAA000OU8
- Product descriptionLY2940680 99%(HPLC)
- Packaging1mg
- Price$15
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000OU8
- Product descriptionLY2940680 99%(HPLC)
- Packaging5mg
- Price$25
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging5MG
- Price$45
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging5MG
- Price$45
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging25MG
- Price$150
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging25MG
- Price$150
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging100MG
- Price$450
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging100MG
- Price$450
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging1G
- Price$1450
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8909
- Product descriptionLY2940680 98%
- Packaging1G
- Price$1450
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberX7613
- Product description4-fluoro-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-2-(trifluoromethyl)benzamide
- Packaging25mg
- Price$254
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0013718
- Product description4-FLUORO-N-METHYL-N-[1-[4-(1-METHYL-1H-PYRAZOL-5-YL)-1-PHTHALAZINYL]-4-PIPERIDINYL]-2-(TRIFLUOROMETHYL)BENZAMIDE 95.00%
- Packaging1MG
- Price$173.25
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0013718
- Product description4-FLUORO-N-METHYL-N-[1-[4-(1-METHYL-1H-PYRAZOL-5-YL)-1-PHTHALAZINYL]-4-PIPERIDINYL]-2-(TRIFLUOROMETHYL)BENZAMIDE 95.00%
- Packaging5MG
- Price$498.43
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8651
- Product descriptionLY2940680
- Packaging50mg
- Price$470
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8651
- Product descriptionLY2940680
- Packaging50mg
- Price$470
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberA8651
- Product descriptionLY2940680
- Packaging200mg
- Price$1386
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA000OU8 | LY2940680 99%(HPLC) | 1mg | $15 | 2026-05-25 | Buy |
| aablocks | AA000OU8 | LY2940680 99%(HPLC) | 5mg | $25 | 2026-05-25 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 5MG | $45 | 2026-05-25 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 5MG | $45 | 2026-05-27 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 25MG | $150 | 2026-05-25 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 25MG | $150 | 2026-05-27 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 100MG | $450 | 2026-05-25 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 100MG | $450 | 2026-05-27 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 1G | $1450 | 2026-05-25 | Buy |
| ACHEMBLOCK | H-8909 | LY2940680 98% | 1G | $1450 | 2026-05-27 | Buy |
| AK Scientific | X7613 | 4-fluoro-N-methyl-N-(1-(4-(1-methyl-1H-pyrazol-5-yl)phthalazin-1-yl)piperidin-4-yl)-2-(trifluoromethyl)benzamide | 25mg | $254 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0013718 | 4-FLUORO-N-METHYL-N-[1-[4-(1-METHYL-1H-PYRAZOL-5-YL)-1-PHTHALAZINYL]-4-PIPERIDINYL]-2-(TRIFLUOROMETHYL)BENZAMIDE 95.00% | 1MG | $173.25 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0013718 | 4-FLUORO-N-METHYL-N-[1-[4-(1-METHYL-1H-PYRAZOL-5-YL)-1-PHTHALAZINYL]-4-PIPERIDINYL]-2-(TRIFLUOROMETHYL)BENZAMIDE 95.00% | 5MG | $498.43 | 2021-12-16 | Buy |
| ApexBio Technology | A8651 | LY2940680 | 50mg | $470 | 2021-12-16 | Buy |
| ApexBio Technology | A8651 | LY2940680 | 50mg | $470 | 2026-05-06 | Buy |
| ApexBio Technology | A8651 | LY2940680 | 200mg | $1386 | 2021-12-16 | Buy |
Properties
Boiling point :703.5±60.0 °C(Predicted)
Density :1.39
storage temp. :Store at -20°C
solubility :insoluble in H2O; ≥5.2 mg/mL in EtOH with ultrasonic; ≥51.3 mg/mL in DMSO with gentle warming and ultrasonic
form :crystalline solid
pka :7.94±0.30(Predicted)
color :White to off-white
Density :1.39
storage temp. :Store at -20°C
solubility :insoluble in H2O; ≥5.2 mg/mL in EtOH with ultrasonic; ≥51.3 mg/mL in DMSO with gentle warming and ultrasonic
form :crystalline solid
pka :7.94±0.30(Predicted)
color :White to off-white
Safety Information
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| Signal word: | Danger | |||||||||||||||||||||
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Description
Smoothened (Smo) is a GPCR-like receptor that, with Patched, mediates hedgehog (Hh) signaling to regulate gene expression through the Gli transcription factors. LY2940680 is an antitumor agent that binds to the human Smo receptor and inhibits Sonic Hh-induced Gli1 expression (IC50 = ~2.4 nM in vitro). The potential anticancer activity of LY2940680 is currently under clinical investigation.More related product prices
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