Mirogabalin
|
- $68 - $3500
- Product name: Mirogabalin
- CAS: 1138245-13-2
- MF: C12H19NO2
- MW: 209.28
- EINECS:-0
- MDL Number:MFCD28411425
- Synonyms:Mirogabalin;[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid;A200-0700;DS5565;A200-0700;2-[(1R,5S,6S)-6-(aminomethyl)-3-ethyl-6-bicyclo[3.2.0]hept-3-enyl]acetic acid;MIROGABALIN; DS-5565;DS 5565;DS-5565;DS5565;Bicyclo[3.2.0]hept-3-ene-6-acetic acid, 6-(aminomethyl)-3-ethyl-, (1R,5S,6S)-
17 prices
Selected condition：
Brand
- AK Scientific
- American Custom Chemicals Corporation
- Biosynth Carbosynth
- Cayman Chemical
- Chemenu
- ChemScene
- DC Chemicals
- TRC
Package
- 1mg
- 2.5mg
- 5MG
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- 100g
- ManufacturerAK Scientific
- Product number4972DP
- Product descriptionMirogabalin
- Packaging10mg
- Price$245
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0028663
- Product descriptionMIROGABALIN 95.00%
- Packaging5MG
- Price$496.06
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBM166964
- Product descriptionMirogabalin
- Packaging10mg
- Price$145
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBM166964
- Product descriptionMirogabalin
- Packaging50mg
- Price$507.5
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number22475
- Product descriptionMirogabalin ≥98%
- Packaging1mg
- Price$68
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number22475
- Product descriptionMirogabalin ≥98%
- Packaging5mg
- Price$152
- Updated2024-03-01
- Buy
- ManufacturerChemenu
- Product numberCM247838
- Product descriptionMirogabalin 98%
- Packaging100g
- Price$3500
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging5mg
- Price$120
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging10mg
- Price$190
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging25mg
- Price$300
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging50mg
- Price$450
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging100mg
- Price$750
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC10013
- Product descriptionMirogabalin >98%
- Packaging100mg
- Price$700
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC10013
- Product descriptionMirogabalin >98%
- Packaging250mg
- Price$1300
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC10013
- Product descriptionMirogabalin >98%
- Packaging1g
- Price$2500
- Updated2021-12-16
- Buy
- ManufacturerTRC
- Product numberM364940
- Product descriptionMirogabalin
- Packaging1mg
- Price$140
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 4972DP | Mirogabalin | 10mg | $245 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0028663 | MIROGABALIN 95.00% | 5MG | $496.06 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BM166964 | Mirogabalin | 10mg | $145 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BM166964 | Mirogabalin | 50mg | $507.5 | 2021-12-16 | Buy |
| Cayman Chemical | 22475 | Mirogabalin ≥98% | 1mg | $68 | 2024-03-01 | Buy |
| Cayman Chemical | 22475 | Mirogabalin ≥98% | 5mg | $152 | 2024-03-01 | Buy |
| Chemenu | CM247838 | Mirogabalin 98% | 100g | $3500 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 5mg | $120 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 10mg | $190 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 25mg | $300 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 50mg | $450 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 100mg | $750 | 2021-12-16 | Buy |
| DC Chemicals | DC10013 | Mirogabalin >98% | 100mg | $700 | 2021-12-16 | Buy |
| DC Chemicals | DC10013 | Mirogabalin >98% | 250mg | $1300 | 2021-12-16 | Buy |
| DC Chemicals | DC10013 | Mirogabalin >98% | 1g | $2500 | 2021-12-16 | Buy |
| TRC | M364940 | Mirogabalin | 1mg | $140 | 2021-12-16 | Buy |
Properties
Boiling point :357.5±15.0 °C(Predicted)
Density :1.104±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF:0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Ethanol:1.25(Max Conc. mg/mL);5.97(Max Conc. mM)
PBS (pH 7.2):0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Water:5.36(Max Conc. mg/mL);25.61(Max Conc. mM) form :A crystalline solid
pka :4.65±0.10(Predicted)
color :Light yellow to light brown
InChI :InChI=1S/C12H19NO2/c1-2-8-3-9-5-12(7-13,6-11(14)15)10(9)4-8/h4,9-10H,2-3,5-7,13H2,1H3,(H,14,15)/t9-,10-,12-/m1/s1
InChIKey :FTBQORVNHOIASH-CKYFFXLPSA-N
SMILES :[C@]12([H])[C@]([H])([C@@](CN)(CC(O)=O)C1)C=C(CC)C2
Density :1.104±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF:0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Ethanol:1.25(Max Conc. mg/mL);5.97(Max Conc. mM)
PBS (pH 7.2):0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Water:5.36(Max Conc. mg/mL);25.61(Max Conc. mM) form :A crystalline solid
pka :4.65±0.10(Predicted)
color :Light yellow to light brown
InChI :InChI=1S/C12H19NO2/c1-2-8-3-9-5-12(7-13,6-11(14)15)10(9)4-8/h4,9-10H,2-3,5-7,13H2,1H3,(H,14,15)/t9-,10-,12-/m1/s1
InChIKey :FTBQORVNHOIASH-CKYFFXLPSA-N
SMILES :[C@]12([H])[C@]([H])([C@@](CN)(CC(O)=O)C1)C=C(CC)C2
Safety Information
| Symbol(GHS): |
|
|||||||||||||||||||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Signal word: | Warning | |||||||||||||||||||||||||||||||||||
| Hazard statements: |
|
|||||||||||||||||||||||||||||||||||
| Precautionary statements: |
|
Description
Mirogabalin is a calcium channel blocker with analgesic effects. It binds to the α2δ-1 and α2δ-2 subunits of voltage-dependent Ca2+ channels. Mirogabalin has potent and sustained analgesic effects (ED50 = 2.5 mg/kg) in rats with diabetes induced by streptozotocin (STZ; ). Mirogabalin does not inhibit activities associated with CNS adverse effects of analgesics, such as rotarod performance (ID50 = 9.4 mg/kg) or locomotor activity (ID50 = 43.9 mg/kg), at its effective dose. Formulations containing mirogabalin are in clinical trials for diabetic peripheral neuropathic pain.Suppliers and manufacturers
Beijing Hope Pharmaceutical Co., Ltd.
Wuhan Circle Star Chem-medical Technology Co.,Ltd
ATK CHEMICAL COMPANY LIMITED
BOC Sciences
HANGZHOU CLAP TECHNOLOGY CO.,LTD
