Mizolastine
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- $21 - $1841
- Product name: Mizolastine
- CAS: 108612-45-9
- MF: C24H25FN6O
- MW: 432.49
- EINECS:1308068-626-2
- MDL Number:MFCD23140913
- Synonyms:4(1h)-pyrimidinone,2-((1-(1-((4-fluorophenyl)methyl)-1h-benzimidazol-2-yl)-4-p ;iperidinyl)methylamino)- ;2-[[1-[1-[(4-fluorophenyl)methyl]benzoimidazol-2-yl]-4-piperidyl]-methyl-amino]-3h-pyrimidin-4-one;MIZOLASTINE;2-[[1-[1-[(4-fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(1H)-pyrimidinone;Mizolastine HCl;2-[[1-[1-(4-fluorobenzyl)benzimidazol-2-yl]-4-piperidyl]-methyl-amino]-1H-pyrimidin-6-one;2-[[1-[1-[(4-fluorophenyl)methyl]benzimidazol-2-yl]piperidin-4-yl]-methyl-amino]-1H-pyrimidin-6-one
49 prices
Selected condition：
Brand
- aablocks
- AHH
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Apolloscientific
- AvaChem
- Cayman Chemical
- Chem-Impex
- ChemScene
- Crysdot
- DC Chemicals
- Matrix Scientific
- Sigma-Aldrich
- TCI Chemical
- TRC
- Usbiological
Package
- 25mg
- 0.1g
- 100mg
- 10mM(in1mLDMSO)
- 5mg
- 10mg
- 50mg
- 200mg
- 250mg
- 500mg
- 1g
- 5g
- 25g
- 100g
- 10 mg
- Manufactureraablocks
- Product numberAA007C3L
- Product description2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone ≥98%
- Packaging200mg
- Price$27
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA007C3L
- Product description2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone ≥98%
- Packaging1g
- Price$56
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA007C3L
- Product description2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone ≥98%
- Packaging5g
- Price$200
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA007C3L
- Product description2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone 98%
- Packaging25g
- Price$807
- Updated2026-05-28
- Buy
- ManufacturerAHH
- Product numberAPI-1754
- Product descriptionMizolastine 97%
- Packaging0.1g
- Price$370
- Updated2026-05-26
- Buy
- ManufacturerAK Scientific
- Product numberI520
- Product descriptionMizolastine 98%
- Packaging5g
- Price$241
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ98981
- Product descriptionMizolastine 95%
- Packaging5g
- Price$180
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10320
- Product descriptionMizolastine >98%,powder
- Packaging100mg
- Price$95
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberI520
- Product descriptionMizolastine 98%
- Packaging1g
- Price$62
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10320
- Product descriptionMizolastine >98%,powder
- Packaging5mg
- Price$22
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ98981
- Product descriptionMizolastine 95%
- Packaging1g
- Price$46
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10320
- Product descriptionMizolastine >98%,powder
- Packaging25mg
- Price$48
- Updated2026-06-04
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0003411
- Product descriptionMIZOLASTINE 95.00%
- Packaging25MG
- Price$160.65
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0003411
- Product descriptionMIZOLASTINE 95.00%
- Packaging100MG
- Price$716.1
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0003411
- Product descriptionMIZOLASTINE 95.00%
- Packaging1G
- Price$1686.3
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1551
- Product descriptionMizolastine
- Packaging10mM(in1mLDMSO)
- Price$50
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA007C3L | 2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone ≥98% | 200mg | $27 | 2026-05-28 | Buy |
| aablocks | AA007C3L | 2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone ≥98% | 1g | $56 | 2026-05-28 | Buy |
| aablocks | AA007C3L | 2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone ≥98% | 5g | $200 | 2026-05-28 | Buy |
| aablocks | AA007C3L | 2-[[1-[1-[(4-Fluorophenyl)methyl]-1H-benzimidazol-2-yl]-4-piperidinyl]methylamino]-4(3H)-pyrimidinone 98% | 25g | $807 | 2026-05-28 | Buy |
| AHH | API-1754 | Mizolastine 97% | 0.1g | $370 | 2026-05-26 | Buy |
| AK Scientific | I520 | Mizolastine 98% | 5g | $241 | 2026-06-04 | Buy |
| AK Scientific | J98981 | Mizolastine 95% | 5g | $180 | 2026-06-04 | Buy |
| AK Scientific | J10320 | Mizolastine >98%,powder | 100mg | $95 | 2026-06-04 | Buy |
| AK Scientific | I520 | Mizolastine 98% | 1g | $62 | 2026-06-04 | Buy |
| AK Scientific | J10320 | Mizolastine >98%,powder | 5mg | $22 | 2026-06-04 | Buy |
| AK Scientific | J98981 | Mizolastine 95% | 1g | $46 | 2026-06-04 | Buy |
| AK Scientific | J10320 | Mizolastine >98%,powder | 25mg | $48 | 2026-06-04 | Buy |
| American Custom Chemicals Corporation | API0003411 | MIZOLASTINE 95.00% | 25MG | $160.65 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0003411 | MIZOLASTINE 95.00% | 100MG | $716.1 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0003411 | MIZOLASTINE 95.00% | 1G | $1686.3 | 2021-12-16 | Buy |
| ApexBio Technology | B1551 | Mizolastine | 10mM(in1mLDMSO) | $50 | 2026-05-06 | Buy |
Properties
Melting point :217°
Density :1.34±0.1 g/cm3(Predicted)
storage temp. :Refrigerator
solubility :Chloroform (Slightly, Heated), DMSO, Methanol (Slightly, Heated)
form :Solid
pka :9.73±0.40(Predicted)
color :White
Merck :14,6221
InChI :1S/C24H25FN6O/c1-29(23-26-13-10-22(32)28-23)19-11-14-30(15-12-19)24-27-20-4-2-3-5-21(20)31(24)16-17-6-8-18(25)9-7-17/h2-10,13,19H,11-12,14-16H2,1H3,(H,26,28,32)
InChIKey :PVLJETXTTWAYEW-UHFFFAOYSA-N
SMILES :C1(N(C2CCN(C3N(CC4=CC=C(F)C=C4)C4=CC=CC=C4N=3)CC2)C)=NC=CC(=O)N1
Density :1.34±0.1 g/cm3(Predicted)
storage temp. :Refrigerator
solubility :Chloroform (Slightly, Heated), DMSO, Methanol (Slightly, Heated)
form :Solid
pka :9.73±0.40(Predicted)
color :White
Merck :14,6221
InChI :1S/C24H25FN6O/c1-29(23-26-13-10-22(32)28-23)19-11-14-30(15-12-19)24-27-20-4-2-3-5-21(20)31(24)16-17-6-8-18(25)9-7-17/h2-10,13,19H,11-12,14-16H2,1H3,(H,26,28,32)
InChIKey :PVLJETXTTWAYEW-UHFFFAOYSA-N
SMILES :C1(N(C2CCN(C3N(CC4=CC=C(F)C=C4)C4=CC=CC=C4N=3)CC2)C)=NC=CC(=O)N1
Safety Information
| Symbol(GHS): |
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| Signal word: | Warning | ||||||||||||||||||||||||||||
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| Precautionary statements: |
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Description
Mizolastine was marketed in Germany and Switzerland as Mizollen for the symptomatic relief of seasonal and perennial allergic rhinoconjunctivitis and urticaria. Mizolastine is a new long-acting, orally active antihistaminic agent with a rapid onset of action ; the two most recent H1 antagonists launched were fexofenadine, metabolite of terfenadine (Sepracor, 1996) and Olopatadine (Kyowa Hakko, 1997). Mizolastine can be prepared in 2 steps from 2-chloro 1- (4-fluorobenzyl)benzimidazole by successive condensations of appropriate amine and thioether. Mizolastine selectively blocks the peripheral H1 receptors (but not the serotonergic, noradrenergic, muscarinic receptors) with a minimal occupancy of brain receptors, and therefore does not elicit any sedative effects. Moreover, Mizolastine does not produce cardiac rhythm disorders which have been associated with certain non-sedating antihistamines in humans.Related product price
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Suppliers and manufacturers
Beijing Jialin Pharmaceutical Co., Ltd.
J & K SCIENTIFIC LTD.
TCI (Shanghai) Development Co., Ltd.
Pure Chemistry Scientific Inc.
Adamas Reagent, Ltd.
LGM Pharma
Chemsky（shanghai）International Co.,Ltd.
Shanghai Sunway Pharmaceutical Technology Co., Ltd
Maya High Purity Chemicals
Dalian Meilun Biotech Co., Ltd.