pristimerin
|
- $65 - $1560
- Product name: pristimerin
- CAS: 1258-84-0
- MF: C30H40O4
- MW: 464.64
- EINECS:251-228-4
- MDL Number:MFCD01711331
- Synonyms:pristimerin;3-Hydroxy-2-oxo-24-nor-D:A-friedoolean-1(10),3,5,7-tetren-29-oic acid methyl ester;Celastrol-methylether;(9β,13α,14β,20α)-3-Hydroxy-9,13-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oicacidmethylester;(9b,13a,14b,20a)-3-Hydroxy-9,13-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tertraen-29-oic acid methyl ester;3-hydroxy-9β,13α-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid, methyl ester;Celastrol methyl ester;Pristimerin(NSC 99281)
45 prices
Selected condition：
Brand
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- AvaChem
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- JR MediChem
- Medical Isotopes, Inc.
- Sigma-Aldrich
- Tocris
- TRC
- Usbiological
Package
- 5MG
- 10
- 1mg
- 10MG
- 20mg
- 25mg
- 50MG
- 100mg
- 1mlx10mM(inDMSO)
- 250mg
- 500mg
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006380
- Product descriptionPristimerin 95.00%
- Packaging5MG
- Price$212.3
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006380
- Product descriptionPristimerin 95.00%
- Packaging10MG
- Price$776.16
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006380
- Product descriptionPristimerin 95.00%
- Packaging50MG
- Price$1515.94
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB7488
- Product descriptionPristimerin
- Packaging50mg
- Price$530
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberB7488
- Product descriptionPristimerin
- Packaging10mg
- Price$130
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB7488
- Product descriptionPristimerin
- Packaging10mg
- Price$130
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberCFN90169
- Product descriptionPristimerin
- Packaging20mg
- Price$128
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2532
- Product descriptionPristimerin
- Packaging25mg
- Price$135
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2532
- Product descriptionPristimerin
- Packaging5mg
- Price$65
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2532
- Product descriptionPristimerin
- Packaging250mg
- Price$790
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2532
- Product descriptionPristimerin
- Packaging100mg
- Price$390
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb594214
- Product descriptionPristimerin
- Packaging20mg
- Price$408
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb1302332
- Product descriptionPristimerin 99.79%(Mayvarybetweenbatches)
- Packaging100mg
- Price$790
- Updated2026-05-06
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb1302332
- Product descriptionPristimerin 99.79%(Mayvarybetweenbatches)
- Packaging50mg
- Price$570
- Updated2026-05-06
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb1302332
- Product descriptionPristimerin 99.79%(Mayvarybetweenbatches)
- Packaging25mg
- Price$340
- Updated2026-05-06
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb1302332
- Product descriptionPristimerin 99.79%(Mayvarybetweenbatches)
- Packaging1mg
- Price$80
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| American Custom Chemicals Corporation | API0006380 | Pristimerin 95.00% | 5MG | $212.3 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0006380 | Pristimerin 95.00% | 10MG | $776.16 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0006380 | Pristimerin 95.00% | 50MG | $1515.94 | 2021-12-16 | Buy |
| ApexBio Technology | B7488 | Pristimerin | 50mg | $530 | 2026-05-06 | Buy |
| ApexBio Technology | B7488 | Pristimerin | 10mg | $130 | 2021-12-16 | Buy |
| ApexBio Technology | B7488 | Pristimerin | 10mg | $130 | 2026-05-06 | Buy |
| Arctom | CFN90169 | Pristimerin | 20mg | $128 | 2021-12-16 | Buy |
| AvaChem | 2532 | Pristimerin | 25mg | $135 | 2021-12-16 | Buy |
| AvaChem | 2532 | Pristimerin | 5mg | $65 | 2021-12-16 | Buy |
| AvaChem | 2532 | Pristimerin | 250mg | $790 | 2021-12-16 | Buy |
| AvaChem | 2532 | Pristimerin | 100mg | $390 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb594214 | Pristimerin | 20mg | $408 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb1302332 | Pristimerin 99.79%(Mayvarybetweenbatches) | 100mg | $790 | 2026-05-06 | Buy |
| Biorbyt Ltd | orb1302332 | Pristimerin 99.79%(Mayvarybetweenbatches) | 50mg | $570 | 2026-05-06 | Buy |
| Biorbyt Ltd | orb1302332 | Pristimerin 99.79%(Mayvarybetweenbatches) | 25mg | $340 | 2026-05-06 | Buy |
| Biorbyt Ltd | orb1302332 | Pristimerin 99.79%(Mayvarybetweenbatches) | 1mg | $80 | 2026-05-06 | Buy |
Properties
Melting point :219.5°C
Boiling point :488.1°C (rough estimate)
Density :1.0271 (rough estimate)
refractive index :1.4800 (estimate)
storage temp. :-20°C
solubility :DMSO: ≥5mg/mL
form :Red solid
pka :8.60±0.70(Predicted)
color :orange
InChIKey :JFACETXYABVHFD-VXTIGNJVNA-N
SMILES :[C@]12(C)CC[C@@]3(C)CC[C@@](C)(C(=O)OC)C[C@@]3([H])[C@]1(C)CC[C@@]1(C)C3=CC(C(O)=C(C)C3=CC=C21)=O |&1:0,4,8,15,17,21,r|
Boiling point :488.1°C (rough estimate)
Density :1.0271 (rough estimate)
refractive index :1.4800 (estimate)
storage temp. :-20°C
solubility :DMSO: ≥5mg/mL
form :Red solid
pka :8.60±0.70(Predicted)
color :orange
InChIKey :JFACETXYABVHFD-VXTIGNJVNA-N
SMILES :[C@]12(C)CC[C@@]3(C)CC[C@@](C)(C(=O)OC)C[C@@]3([H])[C@]1(C)CC[C@@]1(C)C3=CC(C(O)=C(C)C3=CC=C21)=O |&1:0,4,8,15,17,21,r|
Safety Information
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Description
Monoacylglycerol lipase (MAGL) hydrolyzes the endogenous cannabinoid 2-arachidonoyl glycerol (2-AG), terminating its capacity to activate cannabinoid receptors. Pristimerin is a naturally occurring terpenoid that potently inhibits MAGL (IC50 = 93 nM). Its actions are rapid, reversible, and noncompetitive. Pristimerin (1 μM) significantly increases 2-AG levels in isolated rat neurons, indicating that it inhibits endogenous MAGL in cultured cells. Moreover, it does not increase levels of palmitoyl ethanolamide, suggesting that pristimerin does not affect the activity of fatty acid amide hydrolase (FAAH).More related product prices
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Suppliers and manufacturers
Shanghai Zheyan Biotech Co., Ltd.
Chengdu GLP biotechnology Co Ltd
Chengdu Biopurify Phytochemicals Ltd.
CONIER CHEM AND PHARMA LIMITED
Wuhan ChemNorm Biotech Co.,Ltd.
