1197160-78-3 Basic information More..
Product Name:PF-05212384
Synonyms:PF-05212384;PKI587;N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]phenyl]urea;1-(4-(4-(dimethylamino)piperidine-1-carbonyl)phenyl)-3-(4-(4,6-dimorpholino-1,3,5-triazin-2-yl)phenyl)urea;Gedatolisib (PF-05212384, PKI-587);N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]phenyl]urea PF-05212384 (PKI-587);PKI-587 N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]phenyl]urea;PKI-587 ( Gedatolisib )
CAS:1197160-78-3
MF:C32H41N9O4
MW:615.73
EINECS:
Mol File:1197160-78-3.mol
1197160-78-3

Use

Gedatolisib (PF-05212384, PKI-587) is a highly potent dual inhibitor of PI3Kα, PI3Kγ and mTOR with IC50 of 0.4 nM, 5.4 nM and 1.6 nM in cell-free assays, respectively. Phase 2.

PF-05212384 manufacturers

  • Gedatolisib;PKI-587
  • US $200.00-0.00 / g
  • 2021-10-08
  • CAS:1197160-78-3
  • Min. Order: 1g
  • Purity: 98%+
  • Supply Ability: 100kgs
  • PF-05212384
  • US $2.00 / kg
  • 2019-07-06
  • CAS:1197160-78-3
  • Min. Order: 1kg
  • Purity: 99%
  • Supply Ability: 100kg
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