| 1457983-28-6 Basic information More.. |
Product Name: | G-749 | Synonyms: | G-49;G-749 (Free base);G-749;8-Bromo-2-[(1-methyl-4-piperidinyl)amino]-4-[(4-phenoxyphenyl)amino]pyrido[4,3-d]pyrimidin-5(6H)-one;8-Bromo-2-[(1-methyl-4-piperidinyl)amino]-4-[(4-phenoxyphenyl)amino]pyrido[4,3-d]pyrimidin-5(6H)-one G749;G-749, >=98%;8-bromo-2-((1-methylpiperidin-4-yl)amino)-4-((4-phenoxyphenyl)amino)pyrido[4,3-d]pyrimidin-5(6H)-one; Pyrido[4,3-d]pyrimidin-5(6H)-one, 8-bromo-2-[(1-methyl-4-piperidinyl)amino]-4-[(4-phenoxyphenyl)amino]- | CAS: | 1457983-28-6 | MF: | C25H25BrN6O2 | MW: | 521.41 | EINECS: | | Mol File: | 1457983-28-6.mol | |
Use
G-749 is a novel and potent FLT3 inhibitor with IC50 of 0.4 nM, 0.6 nM and 1 nM for FLT3 (WT), FLT3 (D835Y), and Mer, respectively, showing lower potency against other tyrosine kinases.
- NAPHTHOL AS-MX
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- US $1.00 / ASSAYS
- 2019-12-23
- CAS:92-75-1
- Min. Order: 1ASSAYS
- Purity: Min98% HPLC
- Supply Ability: 10t
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1457983-28-6
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