- Rilmenidine
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- $14.00 / 1kg
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2022-12-24
- CAS:54187-04-1
- Min. Order: 1kg
- Purity: 99%
- Supply Ability: 1000kg
- Rilmenidine
-
- $15.00 / 1KG
-
2021-08-12
- CAS:54187-04-1
- Min. Order: 1KG
- Purity: 99%+ HPLC
- Supply Ability: Monthly supply of 1 ton
- Rilmenidine
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- $5.00 / 1KG
-
2020-11-16
- CAS:54187-04-1
- Min. Order: 25KG
- Purity: 99
- Supply Ability: 999
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| | Rilmenidine Basic information |
| Product Name: | Rilmenidine | | Synonyms: | n-(dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine;oxaminozoline;RILMENIDINE;1,1-dicyclopropyl-n-(2-oxazolinyl)-methylamin;2-((dicyclopropylmethyl)imino)-oxazolidin;2-((dicyclopropylmethyl)imino)oxazolidine;2-(dicyclopropylmethylamino)-2-oxazoline;4,5-dihydro-n-(dicyclopropylmethyl)-2-oxazolamin | | CAS: | 54187-04-1 | | MF: | C10H16N2O | | MW: | 180.25 | | EINECS: | 259-021-0 | | Product Categories: | Antihypertensive;Imidazoline binding site | | Mol File: | 54187-04-1.mol |  |
| | Rilmenidine Chemical Properties |
| Melting point | 106-107° | | Boiling point | 355.5±9.0 °C(Predicted) | | density | 1.45±0.1 g/cm3(Predicted) | | storage temp. | Store at -20°C | | solubility | H2O: 7.3 mg/mL | | form | solid | | pka | 7.88±0.50(Predicted) | | color | white | | CAS DataBase Reference | 54187-04-1(CAS DataBase Reference) |
| Safety Statements | 22-24/25 | | WGK Germany | 3 | | RTECS | RP7207400 |
| | Rilmenidine Usage And Synthesis |
| Description | Rilmenidine is a new antihypertensive agent with a selective alphaz-agonist/antagonist
profile, reportedly useful in the management of mild to moderate hypertension. Its
fmt-line indication is possible because of the clear dissociation of its antihypertensive
activity from other neurophannacological effects. | | Chemical Properties | water soluble | | Originator | Servier (France) | | Uses | I1-imidazoline binding site ligand and a2-adrenoceptor agonist, exhibits higher I1 vs. a2 selectivity than clonidine | | Definition | ChEBI: Rilmenidine is an isourea. | | Brand name | Hyperium | | Biological Activity | I 1 -imidazoline binding site selective ligand and α 2 -adrenoceptor agonist. Possesses greater I 1 vs α 2 selectivity than the prototypical compound, clonidine. | | Metabolic pathway | In short-term rat hepatocyte cultures, oxaminozoline is
metabolized and its four metabolites resulting from
oxidation or hydrolysis are identified, three of which
are identical to those reported in vivo. The presence of
an additional minor metabolite in culture may be due
to the higher metabolic rate of oxaminozoline in this
model system. |
| | Rilmenidine Preparation Products And Raw materials |
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