BS 181 Dihydrochloride

BS 181 Dihydrochloride Suppliers list
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Products Intro: Product Name:BS 181 dihydrochloride
CAS:1883548-83-1
Purity:>=99%(HPLC) Package:$183.9/10mg;$770.9/50mg;Bulk package Remarks:99%(HPLC)
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Products Intro: Product Name:BS-181 dihydrochloride
CAS:1883548-83-1
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Company Name: Shanghai Hongye Biotechnology Co. Ltd  
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Products Intro: Product Name:BS 181 dihydrochloride
CAS:1883548-83-1
Purity:>98% Package:1mg;10mg;50mg;100mg;
Company Name: Nantong QuanYi Biotechnology Co., Ltd  
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Products Intro: Product Name:BS-181 dihydrochloride
CAS:1883548-83-1
Purity:98%+ HPLC Package:10mg,500mg,1g,2g,5g,10g,More
Company Name: TargetMol Chemicals Inc.  
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Products Intro: Product Name:BS-181 dihydrochloride
CAS:1883548-83-1
Package:50mg/RMB 17500;10mg/RMB 4200
BS 181 Dihydrochloride Basic information
Product Name:BS 181 Dihydrochloride
Synonyms:BS 181 Dihydrochloride
CAS:1883548-83-1
MF:C22H33ClN6
MW:417
EINECS:
Product Categories:
Mol File:1883548-83-1.mol
BS 181 Dihydrochloride Structure
BS 181 Dihydrochloride Chemical Properties
storage temp. Store at -20°C
solubility Soluble in DMSO
Safety Information
MSDS Information
BS 181 Dihydrochloride Usage And Synthesis
UsesBS 181 Dihydrochloride is a selective cdk7 inhibitor. It promotes cell cycle arrest and apoptosis in a range of cancer cells in vitro and inhibits MCF-7 tumor xenograft growth in mice.
in vivo

BS-181 dihydrochloride (intraperitoneal injection; 10 mg/kg, 20 mg/kg; single dose) is well tolerated in mice without apparent weight altering[1].BS-181 dihydrochloride (intraperitoneal injection; 5 mg/kg or 10 mg/kg twice daily; total daily doses of 10 mg/kg or 20 mg/kg; 14 days) inhibitstumor growth in a dose-dependent manner. Tumor growth exhibits 25% and 50% reduction compared with the control group, for 10 mg/kg/day and 20 mg/kg/day, respectively[1].

Animal Model:7-week old female nu/nu-BALB/c athymic nude mice?with MCF-7 cells[1]
Dosage:5 mg/kg or 10 mg/kg; 10 mg/kg or 20 mg/kg
Administration:Intraperitoneal injection; twice daily or once total daily; 14 days
Result:Inhibited tumor growth significantly.
IC 50CDK7: 21 nM (IC50); CDK2: 880 nM (IC50); CDK5: 3000 nM (IC50); CDK9: 4200 nM (IC50)
storageStore at +4°C
BS 181 Dihydrochloride Preparation Products And Raw materials
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