ChemicalBook > Product Catalog >Biochemical Engineering >Inhibitors >TGF-beta / Smad >PKC inhibitor >GF109203X

GF109203X

GF109203X Suppliers list
Company Name: ATK CHEMICAL COMPANY LIMITED
Tel: +86 21 5161 9050/ 5187 7795
Email: ivan@atkchemical.com
Products Intro: Product Name:GF109203X;G 6850
CAS:133052-90-1
Purity:98% HPLC Package:5MG;10MG;50MG;100MG,1G,5G
Company Name: Biochempartner
Tel: 0086-13720134139
Email: candy@biochempartner.com
Products Intro: Product Name:GF109203X
CAS:133052-90-1
Purity:98% HPLC LCMS Package:10G;20G
Company Name: J & K SCIENTIFIC LTD.  
Tel: 400-666-7788 +86-10-82848833
Email: jkinfo@jkchemical.com;market6@jkchemical.com
Products Intro: Product Name:GF 109203X
CAS:133052-90-1
Package:10Mg,1Mg,5Mg
Company Name: 3B Pharmachem (Wuhan) International Co.,Ltd.  
Tel: 86-21-50328103 * 801、802、803、804 Mobile:18930552037
Email: 3bsc@sina.com
Products Intro: Product Name:GF 109203X;2-[1-(3-DiMethylaMinopropyl)indol-3-yl]-3-(indol-3-yl)MaleiMide
CAS:133052-90-1
Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
Company Name: VDM Biochemicals   
Tel: 0330-2528181
Email: sales@vdmbio.com
Products Intro: Product Name:GF 109203X
CAS:133052-90-1
Purity:>=98%HPLC
GF109203X Basic information
Product Name:GF109203X
Synonyms:InSolution Bisindolylmaleimide I - CAS 133052-90-1 - Calbiochem;GO 6850;GO 6850 HCL;GF 109203X;GF-109203X HCL;GF109203X HYDROCHLORIDE;BISINDOLYLMALEIMIDE;BISINDOLYLMALEIMIDE I
CAS:133052-90-1
MF:C25H24N4O2
MW:412.48
EINECS:
Product Categories:Protein Kinase;inhibitor;TGF-beta/Smad;Inhibitors;Smad;TGF-beta
Mol File:133052-90-1.mol
GF109203X Structure
GF109203X Chemical Properties
Melting point 280℃ (decomposition)
storage temp. 2-8°C
solubility DMSO: ~1 mg/mlsoluble
form Liquid
Water Solubility Insoluble in water.
Safety Information
Hazard Codes Xn
Risk Statements 40-22
Safety Statements 36/37
WGK Germany 3
RTECS UX9590000
MSDS Information
ProviderLanguage
SigmaAldrich English
GF109203X Usage And Synthesis
Biological ActivityVery potent and selective inhibitor of protein kinase C, selective for the α and β 1 isoforms (IC 50 values are 0.0084, 0.0180, 0.210, 0.132, and 5.8 μ M for α , β 1, δ , ε , and ζ isoforms respectively). Selective over MLCK, PKG and PKA (IC 50 values are 0.6, 4.6, and 33 μ M respectively). Potent antagonist at the 5-HT 3 receptor (K i = 29.5 nM). Anti-inflammatory in vivo . Also available as part of the Mixed Kinase Inhibitor Tocriset™ .
GF109203X Preparation Products And Raw materials
Tag:GF109203X(133052-90-1) Related Product Information
BISINDOLYLMALEIMIDE III, HYDROCHLORIDE,BISINDOLYLMALEIMIDE III, HYDROCHLORIDE Bisindolylmaleimide III, HCl BISINDOLYLMALEIMIDE IX METHANESULFONATE BISINDOLYLMALEIMIDE III, ACETATE BISINDOLYLMALEIMIDE IV BISINDOLYLMALEIMIDE VIII ACETATE BISINDOLYLMALEIMIDE IX, METHANESULFONATE,BISINDOLYLMALEIMIDE IX METHANESULPHONATE SALT BISINDOLYLMALEIMIDE III Bisindolylmaleimide I, HCl BISINDOLYLMALEIMIDE VIII ACETATE SALT BISINDOLYLMALEIMIDE V RHODAMINE-CONJUGATED BISINDOLYLMALEIMIDE INHIBITOR BISINDOLYLMALEIMIDE II Bisindolylmaleimide Inhibitor Set BISINDOLYLMALEIMIDE VI BISINDOLYLMALEIMIDE X, HCL,BISINDOLYLMALEIMIDE X HYDROCHLORIDE,BISINDOLYLMALEIMIDE X HYDROCHLORIDE GO 6983 GF109203X