hTG2 inhibitor VA4 (VA4)

hTG2 inhibitor VA4 (VA4) Suppliers list

Company Name:	TargetMol Chemicals Inc.
Tel:	+17819995354
Email:	marketing@targetmol.com
Products Intro:	Product Name:VA4 TG2 inhibitor CAS:2088001-23-2 Package:100mg;2500USD\|25mg;1520USD\|50mg;1980USD

Company Name:	TargetMol Chemicals Inc.
Tel:	15002134094
Email:	marketing@targetmol.cn
Products Intro:	Product Name:VA4 TG2 inhibitor CAS:2088001-23-2 Package:100mg/RMB 17500;25mg/RMB 10600;50mg/RMB 13800

hTG2 inhibitor VA4 (VA4) manufacturers

hTG2 inhibitor VA4 (VA4) Basic information

Product Name:	hTG2 inhibitor VA4 (VA4)
Synonyms:	hTG2 inhibitor VA4 (VA4);VA4;Carbamic acid, N-[(1S)-1-[[4-[[5-(dimethylamino)-1-naphthalenyl]sulfonyl]-1-piperazinyl]carbonyl]-5-[(1-oxo-2-propen-1-yl)amino]pentyl]-, phenylmethyl ester;Benzyl(S)-(6-acrylamido-1-(4-((5-(dimethylamino)naphthalen-1-yl)sulfonyl)piperazin-1-yl)-1-oxohexan-2-yl)carbamate;VA4 TG2 inhibitor
CAS:	2088001-23-2
MF:	C33H41N5O6S
MW:	635.77
EINECS:
Product Categories:
Mol File:	2088001-23-2.mol

hTG2 inhibitor VA4 (VA4) Chemical Properties

Safety Information

MSDS Information

hTG2 inhibitor VA4 (VA4) Usage And Synthesis

Description	VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.
Uses	hTG2 inhibitor VA4 (compound VA4) is an irreversible Type 2 transglutaminase (TG2) inhibitor. hTG2 inhibitor VA4 reacts exclusively at the TG2 transamidase site, inhibits both transamidase and GTP-binding activities[1].
References	[1] Kerr C, et al. Transamidase site-targeted agents alter the conformation of the transglutaminase cancer stem cell survival protein to reduce GTP binding activity and cancer stem cell survival. Oncogene. 2017 May 25;36(21):2981-2990. DOI:10.1038/onc.2016.452

hTG2 inhibitor VA4 (VA4) Preparation Products And Raw materials

Tag:hTG2 inhibitor VA4 (VA4)(2088001-23-2) Related Product Information

HomePage | Member Companies | Advertising | Contact us | Previous WebSite | MSDS | CAS Index | CAS DataBase | Privacy | Terms | About Us
All products displayed on this website are only for non-medical purposes such as industrial applications or scientific research, and cannot be used for clinical diagnosis or treatment of humans or animals. They are not medicinal or edible.
According to relevant laws and regulations and the regulations of this website, units or individuals who purchase hazardous materials should obtain valid qualifications and qualification conditions.