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| 5-METHOXYGRAMINE Basic information |
| 5-METHOXYGRAMINE Chemical Properties |
Melting point | 123-126 °C (lit.) | Boiling point | 342.77°C (rough estimate) | density | 1.0565 (rough estimate) | refractive index | 1.6000 (estimate) | storage temp. | Refrigerator (+4°C) | pka | 16.70±0.30(Predicted) | BRN | 170533 | CAS DataBase Reference | 16620-52-3(CAS DataBase Reference) |
Hazard Codes | C,Xi | Risk Statements | 34-22 | Safety Statements | 22-24/25 | WGK Germany | 3 | RTECS | NL7700000 | F | 10 | HS Code | 29339900 | Toxicity | mouse,LD50,intraperitoneal,130mg/kg (130mg/kg),Psychopharmacologia Vol. 16, Pg. 385, 1970. |
| 5-METHOXYGRAMINE Usage And Synthesis |
Chemical Properties | white to almost white crystalline powder | Uses | - Reactant for preparation of dopamine D2 receptor antagonists
- Reactant for asymmetric preparation of ethenyl(tetrahydro)carbazoledicarboxylates via gold(I)-catalyzed intramolecular Friedel-Crafts allylic alkylation reaction
- Reactant for preparation of N-substituted 3-aryl-8-azabicyclo[3.2.1]octan-3-ols as dopamine D2-like receptor ligands
- Reactant for preparation of substituted N-trimethoxybenzoyl indoles, indolines, and a tetrahydroquinoline via N-aroylation with trimethoxybenzoyl chloride or anhydride as antitubulin agents
- Reactant for preparation of indolylmethanesulfonamide and its methoxy derivatives
| Uses | • ;Reactant for preparation of dopamine D2 receptor antagonists1• ;Reactant for asymmetric preparation of ethenyl(tetrahydro)carbazoledicarboxylates via gold(I)-catalyzed intramolecular Friedel-Crafts allylic alkylation reaction2• ;Reactant for preparation of N-substituted 3-aryl-8-azabicyclo[3.2.1]octan-3-ols as dopamine D2-like receptor ligands3• ;Reactant for preparation of substituted N-trimethoxybenzoyl indoles, indolines, and a tetrahydroquinoline via N-aroylation with trimethoxybenzoyl chloride or anhydride as antitubulin agents4• ;Reactant for preparation of in |
| 5-METHOXYGRAMINE Preparation Products And Raw materials |
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