| Company Name: | 
                                
                                    Shanghai Aladdin Bio-Chem Technology Co.,LTD  
                                 | 
                             
                            
                                | Tel: | 
                                400-6206333 13167063860 | 
                             
                            
                                | Email: | 
                                anhua.mao@aladdin-e.com | 
                             
                            
                                | Products Intro: | 
                                
                                    Product Name:Apatinib-d8 Hydrochloride CAS:2468771-44-8 Purity:98%,95atom%D  Package:1mg/RMB 4184.90;5mg/RMB 4399.90
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                                | Company Name: | 
                                
                                    LGC Science (Shanghai) Ltd.  
                                 | 
                             
                            
                                | Tel: | 
                                 17717235263 | 
                             
                            
                                | Email: | 
                                cindy.yang@lgcgroup.com | 
                             
                            
                                | Products Intro: | 
                                
                                    Product Name:Apatinib-d8 Hydrochloride CAS:2468771-44-8 Purity:具体纯度,见COA  Package:50mg  Remarks:TRC-A726152
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                                | Company Name: | 
                                
                                    TargetMol Chemicals Inc.  
                                 | 
                             
                            
                                | Tel: | 
                                 15002134094 | 
                             
                            
                                | Email: | 
                                marketing@targetmol.cn | 
                             
                            
                                | Products Intro: | 
                                
                                    Product Name:Apatinib-d8 Hydrochloride CAS:2468771-44-8   Package:1mg;5mg
                                 | 
                             
                        
                     
                    
                    
                        
                            
                                | Company Name: | 
                                
                                    SHANGHAI ZZBIO CO., LTD.  
                                 | 
                             
                            
                                | Tel: | 
                                15102117276 19921389125 | 
                             
                            
                                | Email: | 
                                tech@zzbioco.com | 
                             
                            
                                | Products Intro: | 
                                
                                    Product Name:Apatinib-d8 Hydrochlorid CAS:2468771-44-8 Purity:0.95  Package:5mg;
                                 | 
                             
                        
                     
                     
                
              
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                 |  | Apatinib-d8 Hydrochloride Basic information |  
  
                 |  | Apatinib-d8 Hydrochloride Chemical Properties |  
 | Melting point  | >192°C (dec.) |  | storage temp.  | Refrigerator |  | solubility  | DMSO (Slightly), Methanol (Slightly) |  | form  | Solid |  | color  | Off-White to Pale Yellow |  
  
                
                
                 |  | Apatinib-d8 Hydrochloride Usage And Synthesis |  
 | Uses | Labelled Apatinib (A726150). Apatinib is an orally available, small molecule multitargeted tyrosine kinase inhibitor. Apatinib selectively inhibits the vascular endothelial growth factor receptor-2 (V
EGFR2). Apatinib functions by inhibiting VEGF-mediated endothelial cell migration and proliferation thus blocking new blood vessel formation in tumor tissue. Recent studies have shown that Apatinib e
nhances the efficacy of conventional chemotherapeutical drugs in side population (SP) cells and ABCB1-overexpressing leukemia cells. |  
  
                 |  | Apatinib-d8 Hydrochloride Preparation Products And Raw materials |  
  
                
                 
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