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| | PIRENPERONE Basic information |
| Product Name: | PIRENPERONE | | Synonyms: | PIRENPERONE (R-47,465) >97% SEROTONIN 5- HT2 ANTAG;R-47,465, 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrido-[1,2-a] pyrimidin-4-one;3-[2-[4-(4-Fluorobenzoyl)piperidino]ethyl]-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one;3-[2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one;3-(2-(4-(4-Fluorobenzoyl)piperidin-1-yl)ethyl)-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one;4H-Pyrido[1,2-a]pyrimidin-4-one,3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-;R 47465,anxiolytic activity,Pirenperone,5-HT Receptor,Inhibitor,R47465,inhibit,5-hydroxytryptamine Receptor,Serotonin Receptor,R-47465;PIRENPERONE | | CAS: | 75444-65-4 | | MF: | C23H24FN3O2 | | MW: | 393.45 | | EINECS: | 278-213-5 | | Product Categories: | ADALAT | | Mol File: | 75444-65-4.mol |  |
| | PIRENPERONE Chemical Properties |
| Boiling point | 556.3±60.0 °C(Predicted) | | density | 1.26±0.1 g/cm3(Predicted) | | storage temp. | Store at -20°C | | solubility | 0.1 M HCl: 11 mg/mL | | form | solid | | pka | 7.91±0.10(Predicted) | | color | light yellow | | Water Solubility | Water: Insoluble |
| | PIRENPERONE Usage And Synthesis |
| Uses | antianginal, antihypertensive | | Uses | 5-HT2 antagonist | | Uses | Pirenperone is a 5-HT2 serotonin receptor antagonist. Pirenperone also increases phosphorylation in human glioma cells by inhibiting cellular gap junctions. | | Definition | ChEBI: 3-[2-[4-[(4-fluorophenyl)-oxomethyl]-1-piperidinyl]ethyl]-2-methyl-4-pyrido[1,2-a]pyrimidinone is an aromatic ketone. |
| | PIRENPERONE Preparation Products And Raw materials |
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