- JTC 801
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- $9.80 / 1.79999995231628KG
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2020-01-13
- CAS:244218-51-7
- Min. Order: 1g
- Purity: ≥99%
- Supply Ability: 100kg
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| JTC 801 Basic information |
Product Name: | JTC 801 | Synonyms: | JTC 801;N-(4-Amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]benzamidehydrochloride;N-(4-Amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]benzamide monohydrochloride;JTC 801 HCl;JTC-801 hydrochloride;JTC-801/JTC801;N-(4-AMino-2-Methyl-quinolin-6-yl)-2-(4-ethyl-phenoxyMethyl)-benzaMide hydrochloride;Benzamide,N-(4-amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]-, hydrochloride | CAS: | 244218-51-7 | MF: | C26H25N3O2.ClH | MW: | 447.963 | EINECS: | | Product Categories: | Inhibitors | Mol File: | 244218-51-7.mol | |
| JTC 801 Chemical Properties |
Melting point | 235℃ | storage temp. | Inert atmosphere,2-8°C | solubility | DMSO: ≥20mg/mL | form | powder | color | tan | InChIKey | NQLIYKXNAXKMBL-UHFFFAOYSA-N |
Hazard Codes | Xi | Risk Statements | 36 | Safety Statements | 26 | WGK Germany | 1 |
| JTC 801 Usage And Synthesis |
Uses | JTC 801 is a novel opioid receptor-like1 (ORL1) receptor antagonist. | Biological Activity | High affinity, selective NOP receptor antagonist (K i = 8.2 nM). Displays approximately 12.5-, 129- and 1055-fold selectivity over human μ -, κ - and δ -opioid receptors respectively. In vivo shows anti-nociceptive effects in acute pain models. Orally active. | storage | Desiccate at RT |
| JTC 801 Preparation Products And Raw materials |
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