AR-A 2 NEW
| Price | $1670 | $2180 | $2800 |
| Package | 25mg | 50mg | 100mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-08-22 |
Product Details
| Product Name: AR-A 2 | CAS No.: 220051-79-6 |
| Supply Ability: 10g | Release date: 2025/08/22 |
Product Introduction
Bioactivity
| Name | AR-A 2 |
| Description | AR-A 2 is a selective 5-HT1B receptor antagonist with high affinity to guinea pig cortex 5-HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM), exhibiting a 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM). |
| In vitro | AR-A 2 (AR-A000002) is a selective 5-HT1B receptor antagonist, exhibiting an EC50 of 4.5 nM for the guinea pig 5-HT1B receptor. It also binds to the rat cortical 5HT1B/1D receptor (Ki: 20 nM), rat cortex 5-HT2A receptor (Ki: 339 nM), rat hippocampus 5-HT1A receptor (Ki: 3070 nM), and shows affinity for dopamine D2 (Ki: 330 nM) and α1-adrenoceptors (Ki: 490 nM). |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Keywords | α1-adrenoceptor | recombinant guinea pig 5-HT1B receptor | Rat hippocampus 5-HT1A receptor | rat cortical 5HT1B/1D receptor | rat cortex 5-HT2A receptor | guinea pig cortex 5HT1B/1D | guinea pig 5-HT1D receptor | guinea pig 5-HT1B receptor | dopamine D2 | AR-A-000002 | AR-A000002 | AR-A 2 | ARA 2 | AR A 2 |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, Massachusetts, USA
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