Product Details
| Product Name:
ESI-05 |
CAS No.:
5184-64-5 |
| Purity:
98.00% |
Supply Ability:
10g |
| Release date:
2025/12/09 |
Product Introduction
Bioactivity
| Name | ESI-05 |
| Description | ESI-05 (NSC-116966) is a specific EPAC2 (exchange protein directly activated by cAMP 2) antagonist (IC50: 0.4 μM). ESI-05 inhibits cAMP-mediated activation of EPAC2, as well as EAPC2, mediated Rap1 activation. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | DMSO : 83.33 mg/mL (303.7 mM), Sonication is recommended.
10% DMSO+90% Corn Oil : 3.3 mg/mL (12.03 mM), Sonication is recommeded.
|
| Keywords | NSC-116966 | NSC116966 | neurological disorders | mono- acylglycerol acyltransferase | Intracranial hemorrhage (ICH) | insulin secretion | Inhibitor | inhibit | GEF | exchange proteins directly activated by cAMP 2 (EPAC2) | ESI-05 | ESI05 | ESI 05 | EPAC2 | Diglyceride acyltransferase | Diacylglycerol acyltransferase | diabetes | cAMP | Acyltransferase | acyl-CoA:cholesterol acyltransferase |
| Inhibitors Related | Xanthohumol | Lecimibide | OSMI-3 | Bithionol | Cyclandelate | Eldacimibe | YM17E | 2-Furoic acid | Torbafylline | 2-PCCA hydrochloride | Eflucimibe | PF-04620110 |
| Related Compound Libraries | Target-Focused Phenotypic Screening Library | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Inhibitor Library | NO PAINS Compound Library | Bioactive Compounds Library Max | GPCR Compound Library | Anti-Cancer Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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Recommended supplier
| Product name |
Price |
|
Suppliers |
Update time |
|
|
$51.00/1mg |
VIP4Y
|
TargetMol Chemicals Inc.
|
2025-12-05 |
|
|
$1520.00/25mg |
VIP2Y
|
TargetMol Chemicals Inc.
|
2025-10-27 |
|
|
$0.00/10mg |
VIP2Y
|
Xian confluore Biological Technology Co., Ltd.
|
2024-04-01 |
United States