GSK 525768A NEW
| Price | $198 | $347 | $1170 |
| Package | 2mg | 5mg | 25mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-07-21 |
Product Details
| Product Name: GSK 525768A | CAS No.: 1260530-25-3 |
| Supply Ability: 10g | Release date: 2025/07/21 |
Product Introduction
Bioactivity
| Name | GSK 525768A |
| Description | GSK 525768A, the inactive enantiomer of GSK525762A, exhibits no activity towards BET. |
| In vitro | GSK 525768A interacts with the protein's module by establishing hydrogen bonds with the conserved asparagine residue, effectively mimicking the acetylated lysine's binding mechanism. This interaction leads to the compound's binding deeper within the acetylated lysine's binding site, all the while preserving the position of conserved water molecules in the acetyl-lysine binding cavity's base. GSK 525768A exhibits no activity towards BET and is identified as the (R)-enantiomer of GSK525762A. Contrasting its counterpart, GSK525762A, which influences the regulation of apolipoprotein A1 (APOA1) levels in liver cell assays, GSK 525768A does not impact APOA1 release, highlighting a distinctive functional divergence between the two enantiomers. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | DMSO : 100 mg/mL (235.9 mM), Sonication is recommended. |
| Keywords | GSK 525768A |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, Massachusetts, USA
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