Product Details
| Product Name:
ST4206 |
CAS No.:
1246018-36-9 |
| Supply Ability:
10g |
Release date:
2025/08/22 |
Product Introduction
Bioactivity
| Name | ST4206 |
| Description | ST4206 is an antagonist of adenosine A2A. For adenosine A2A receptor and adenosine A1 receptor, the Kis values are 12 nM and 197 nM , respectively. |
| In vitro | ST4206 inhibits agonist-induced cAMP accumulation with an IC50 of 990 nM [1]. |
| In vivo | ST4206, administered orally at doses of 10, 20, and 40 mg/kg, counteracts haloperidol-induced catalepsy and enhances motor activity in mice in a dose-dependent fashion. At dosages of 20 and 40 mg/kg, the compound markedly augments the number of contralateral turns in rats triggered by l-DOPA[1]. Demonstrating oral efficacy at concentrations of 10, 20, and 40 mg/kg, ST4206 effectively mitigates haloperidol-induced catalepsy in mice[2]. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Keywords | ST-4206 | ST4206 | ST 4206 | adenosine A2A receptor | adenosine A1 receptor |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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Recommended supplier
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$2380.00/50mg |
VIP4Y
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TargetMol Chemicals Inc.
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2025-07-16 |
United States