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成都先导药物开发股份有限公司

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  •       成都先导药物开发股份有限公司(上海证券交易所股票代码:688222.SH,股票名称:成都先导)致力于打造全球一流的创新型生物医药企业,贡献于更好的人类生命健康。公司聚焦小分子及核酸新药的发现与优化,依托DNA编码化合物库技术(包括DEL库的设计、合成和筛选及拓展应用)、基于分子片段和三维结构信息的药物设计技术(FBDD/SBDD)、核酸新药研发相关技术(STO)、靶向蛋白降解相关技术(TPD)等四个核心技术平台及公司其他关键新药研发能力(药化、计算科学、生物评价、药学研究等),打造国际领先的新药发现与优化研发体系,通过新药研发服务、不同阶段在研项目转让以及远期的药物上市等多元化的商业模式,为医药工业输出不同阶段的新分子实体,以期最终为全球未满足的临床需求提供创新药治疗方案。成都先导自创立以来始终致力于核心技术——DNA编码化合物库(DEL)技术的开发、应用和升级,是DEL技术领域的领先者之一,截至2021年末,公司的DNA编码化合物库小分子种类已突破12,000亿,是全球目前已知的化合物骨架种类最多规模最大的实体小分子化合物库。成都先导成立于2012年,总部位于中国成都,在英国剑桥、美国休斯顿设有子公司。公司业务遍布北美、欧洲、亚洲、非洲及大洋洲等,现已与多家国际著名制药公司、生物技术公司、化学公司、基金会以及科研机构建立合作。 获取更多信息,请致电+86-28-85197385,+1-508-840-9646或访问www.hitgen.com。 媒体查询:media@hitgen.com 投资者咨询:investors@hitgen.com 商务开发:bd@hitgen.com
英文名称 中文名称 CAS号 操作
4-(4-bromophenoxy)-1-(tert-butoxycarbonyl)piperidine-4-carboxylic acid 4-(4-溴苯氧基)-1-(叔丁氧基羰基)哌啶-4-羧酸 1159835-30-9 详细
2-((bis(4-methoxyphenyl)(phenyl)methoxy)methyl)-6-(2,2,2-trifluoroacetamido)hexyl (2-cyanoethyl) diisopropylphosphoramidite AMINO-MODIFIER C7 CE PHOSPHORAMIDITE 详细
2-(5-bromo-3-(methoxycarbonyl)-1H-indol-1-yl)acetic acid 详细
2-(2-(2-(bis(4-methoxyphenyl)(phenyl)methoxy)ethoxy)ethoxy)ethyl (2-cyanoethyl) diisopropylphosphoramidite SPACER-9 CEP 146668-73-7 详细
(S)-1- (4, 4'-dimethoxytrityl)-3-thymidine-2-cyanoethyl Phosphoramidite T-(S)-GNA phosphoramidite 168332-13-6 详细
N6-benzoyl- (S)- 1- (4, 4'-dimethoxytrityl)-3-adenosine-2-cyanoethyl Phosphoramidite N6-Bz-A-(S)-GNA phosphoramidite 851050-24-3 详细
2'OC16-G(iBu) phosphoramidite DMTR-2'-O-C16-RG(IBU)-3'-CE-PHOSPHORAMIDITE 2382942-32-5 详细
3-[[(2R,3S)-3-[bis(4-methoxyphenyl)-phenylmethoxy]oxolan-2-yl]methoxy-[di(propan-2-yl)amino]phosphanyl]oxypropanenitrile invAb phosphoramidite 401813-16-9 详细
N-(9-((2R,3R,4R,5R)-4-((tert-butyldimethylsilyl)oxy)-5-((R)-cyclopropyl(hydroxy)methyl)-3-methoxytetrahydrofuran-2-yl)-9H-purin-6-yl)benzamide 详细
(2S,4R)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4-(2-(tert-butoxy)-2-oxoethoxy)pyrrolidine-2-carboxylic acid 详细
2-(2-chloro-4-fluoro-5-nitrophenyl)acetic acid 详细
pLNAAprG PLNAAPRG 详细
TNA-G phosphoramidite TNA-G PHOSPHORAMIDITE 详细
N6-benzoyl-5'-O-(4, 4'-dimethoxytrityl)-2'-O-4'-C-Locked-adenosine-3'-cyanoethyl Phosphoramidite LNA-A(Bz) phosphoramidite 206055-79-0 详细
TNA-T phosphoramidite TNA-T PHOSPHORAMIDITE 325683-94-1 详细
UNA-C(Ac) phosphoramidite 1120329-56-7 详细
methyl (2R,4S)-4-azidopyrrolidine-2-carboxylate hydrochloride 详细
(2R,3R)-1-(tert-butoxycarbonyl)-3-(4-iodophenyl)pyrrolidine-2-carboxylic acid 详细
N4-benzoyl-5-methyl-5'-O-(4, 4'-dimethoxytrityl)-2'-O-4'-C-Locked-cytidine-3'-cyanoethyl Phosphoramidite LNA-5mC(Bz) phosphoramidite 206055-82-5 详细
2-(5-bromo-3-(methoxycarbonyl)-2-oxopyridin-1(2H)-yl)acetic acid 详细
4-bromo-3-(methoxycarbonyl)benzoic acid 详细
(S)-1- (4, 4'-dimethoxytrityl)-3-uridine-2-cyanoethyl Phosphoramidite U-(S)-GNA phosphoramidite 494784-15-5 详细
N1,N3,N5-tris(3-(didocecylamino)propyl)benzene-1,3,5-tricarboxamide TT3-LLN 1821214-50-9 详细
{(2R,3S)-3-[Bis-(4-methoxy-phenyl)-phenyl-methoxy]-tetrahydro-furan-2-ylmethoxy}-tert-butyl-dimethyl-silane 401813-07-8 详细
5'-(4,4'-dimethoxytrityl)-2'-benzoyl-2',3'-seco-uridine-3’-cyanoethyl Phosphoramidite UNA-U phosphoramidite 1120329-48-7 详细
2'OC16-U phosphoramidite DMTR-2'-O-C16-RU-3'-CE-PHOSPHORAMIDITE 2382942-83-6 详细
5-OBz-dC(Bz) Phosphoramidite 5-OBZ-DC(BZ) PHOSPHORAMIDITE 197579-70-7 详细
(3-fluoro-4-nitrobenzyl)-L-proline 详细
((2R,3R)-3-(bis(4-methoxyphenyl)(phenyl)methoxy)tetrahydrofuran-2-yl)methanol 详细
deoxyribavirin phosphoramidite DEOXYRIBAVIRIN PHOSPHORAMIDITE 详细
2'OC16-A(Bz) phosphoramidite DMTR-2'-O-C16-RA(BZ)-3'-CE -PHOSPHORAMIDITE 2382942-35-8 详细
3-((5-bromo-3-formylpyridin-2-yl)(methyl)amino)propanoic acid 详细
2-(4-(tert-butoxycarbonyl)piperazin-1-yl)-6-chloroisonicotinic acid 详细
N2-isobutyryl- (S)- 1- (4, 4'-dimethoxytrityl)-3-Guanosine-2-cyanoethyl Phosphoramidite N2-iBu-G-(S)-GNA phosphoramidite 182625-68-9 详细
N2-dimethylformamidine-5'-O-(4, 4'-dimethoxytrityl)-2'-O-4'-C-Locked-Guanosine-3'-cyanoethyl Phosphoramidite LNA-G(dmf) phosphoramidite 详细
6-bromohexyl phosphoramidite 6-BROMOHEXYL PHOSPHORAMIDITE 956093-29-1 详细
2-(((3R,5S)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-5-(azidomethyl)pyrrolidin-3-yl)oxy)acetic acid 详细
(((2R,3R)-3-(bis(4-methoxyphenyl)(phenyl)methoxy)tetrahydrofuran-2-yl)methoxy)(tert-butyl)dimethylsilane 详细
2-(((9H-fluoren-9-yl)methoxy)carbonyl)-8-(tert-butoxycarbonyl)-2,8-diazaspiro[4.5]decane-4-carboxylic acid 2-(((9H-芴-9-基)甲氧基)羰基)-8-(叔-丁氧羰基)-2,8-二氮杂螺[4.5]癸烷-4-羧酸 详细
Tocopherol phosphoramidite TOCOPHEROL PHOSPHORAMIDITE 1772522-16-3 详细
5'-O-(4, 4'-dimethoxytrityl)-2'-O-4'-C-Locked-thymidine-3'-cyanoethyl Phosphoramidite LNA-T phosphoramidite 206055-75-6 详细
dSpacer CE Phosphoramidite 1,4-脱水-5-O-[二(4-甲氧基苯基)苯基甲基]-2-脱氧-D-赤式-戊糖醇 2-氰基乙基 二(异丙基)氨基亚磷酸酯 129821-76-7 详细
N6-benzoyl-5'-(4,4'-dimethoxytrityl)-2'-benzoyl-2',3'-seco-adenosine-3’-cyanoethyl Phosphoramidite UNA-A(Bz) phosphoramidite 1120329-52-3 详细
1-(1-(tert-butoxycarbonyl)azetidin-3-yl)-3-formyl-1H-indole-4-carboxylic acid 详细
Ribavirin phosphoramidite RIBAVIRIN PHOSPHORAMIDITE 详细
2-((2-(Bis(4-methoxyphenyl)(phenyl)methoxy)ethyl)sulfonyl)ethyl(2-cyanoethyl)diisopropylphosphoramidite 5‘ 磷酸化单体 108783-02-4 详细
N4-acetyl-(S)-1- (4, 4'-dimethoxytrityl)-3-cytidine-2-cyanoethyl Phosphoramidite N4-Ac-C-(S)-GNA phosphoramidite 1159174-80-7 详细
pAmpG 2′-O-甲基-5′-O-膦酰基腺苷酰基-(3′→5′)-鸟苷 2638447-50-2 详细
TNA-O6-DPC-G phosphoramidite TNA-O6-DPC-G phosphoramidite 325683-97-4 详细
N-(9-((2R,3R,4R,5R)-4-((tert-butyldimethylsilyl)oxy)-5-((S)-cyclopropyl(hydroxy)methyl)-3-methoxytetrahydrofuran-2-yl)-9H-purin-6-yl)benzamide 详细
2-(6-bromo-3-formyl-1H-indol-1-yl)acetic acid 详细
(2S,4S)-1-(tert-butoxycarbonyl)-4-(4-iodophenoxy)pyrrolidine-2-carboxylic acid 详细
1,1'-((2-(4-(2-((2-(bis(2-hydroxydodecyl)amino)ethyl)(2-hydroxydodecyl)amino)ethyl)piperazin-1-yl)ethyl)azanediyl)bis(dodecan-2-ol) C12-200 1220890-25-4 详细
TNA-C phosphoramidite DMTR-TNA-C(BZ)-AMIDITE 325683-96-3 详细
2'OC16-C(Ac) phosphoramidite DMTR-2'-O-C16-RC(AC)-3'- CE-PHOSPHORAMIDITE 2382942-38-1 详细
TNA-A(Bz) phosphoramidite TNA-A(BZ) PHOSPHORAMIDITE 325683-93-0 详细
(2R,5R,6R)-6-(((((9H-fluoren-9-yl)methoxy)carbonyl)amino)methyl)-5-azidotetrahydro-2H-pyran-2-carboxylic acid 详细
6-(tert-butoxycarbonyl)-2-(methoxycarbonyl)-6-azaspiro[3.4]octane-8-carboxylic acid 详细
N2-isobutyryl-5'-(4,4'-dimethoxytrityl)-2'-benzoyl-2',3'-seco-guanosine-3’-cyanoethyl Phosphoramidite UNA-G(iBu) phosphoramidite 1120329-61-4 详细
N-(9-((2R,3R,4R,5R)-4-((tert-butyldimethylsilyl)oxy)-5-((S)-2-cyclopropyl-1-hydroxyethyl)-3-methoxytetrahydrofuran-2-yl)-9H-purin-6-yl)benzamide 详细
N-(9-((2R,3R,4R,5R)-4-((tert-butyldimethylsilyl)oxy)-5-((R)-2-cyclopropyl-1-hydroxyethyl)-3-methoxytetrahydrofuran-2-yl)-9H-purin-6-yl)benzamide 详细
1-{2'-O-[(4",4"'-dimethoxytriphenyl)methyl]-α-L-threofuranosyl}uracil TNA-U 537690-78-1 详细
产品总数:62 产品页码:
1

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