中文名:AGI-5198,突变体异柠檬酸脱氢酶1(mIDH1)的有效抑制剂
英文名:AGI-5198
英文别名:AGI-5198|1355326-35-0|IDH-C35|N-cyclohexyl-2-(N-(3-fluorophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido)-2-(o-tolyl)acetamide|AGI 5198|N-cyclohexyl-2-(3-fluoro-N-[2-(2-methylimidazol-1-yl)acetyl]anilino)-2-(2-methylphenyl)acetamide|N-cyclohexyl-2-(N-(3-fl
纯度:≥98%
货号:A126546
包装:100mg、25mg、5mg
Cas号:1355326-35-0
存储温度:-20°C储存
产品介绍:
AGI-5198 is the first highly potent and selective inhibitor of IDH1 R132H/R132C mutants with IC50 of 0.07 μM/0.16 μM.AGI-5198(IDH C35)是剂量依赖的R132H-IDH1抑制剂
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