| Identification | Back Directory | [Name]
Butanedioic acid, 1-[7-bromo-5-(2-chlorophenyl)-2,3-dihydro-2-oxo-1H-1,4-benzodiazepin-3-yl] ester | [CAS]
172986-25-3 | [Synonyms]
Cinazepam
1-[7-bromo-5-(2-chlorophenyl)-2,3-dihydro-2-oxo-1H-1,4-benzodiazepin-3-yl] ester, butanedioic acid
Butanedioic acid, 1-[7-bromo-5-(2-chlorophenyl)-2,3-dihydro-2-oxo-1H-1,4-benzodiazepin-3-yl] ester | [Molecular Formula]
C19H14BrClN2O5 | [MOL File]
172986-25-3.mol | [Molecular Weight]
465.68 |
| Chemical Properties | Back Directory | [Boiling point ]
658.4±55.0 °C(Predicted) | [density ]
1.66±0.1 g/cm3(Predicted) | [solubility ]
DMF: 15 mg/ml; DMF:PBS (pH 7.2) (1:9): 0.1 mg/ml; DMSO: 10 mg/ml; Ethanol: 0.2 mg/ml | [form ]
A crystalline solid | [pka]
4.25±0.17(Predicted) |
| Hazard Information | Back Directory | [Description]
Cinazepam is an analytical reference standard categorized as a benzodiazepine. Cinazepam is a prodrug form of 3-hydroxy phenazepam that has anxiolytic and sedative properties. This product is intended for research and forensic applications. | [Uses]
Cinazepam has been used in the novel combination therapy for anxiety disorders, epilepsy, and pain comprising GABA agonist and inhibitor. | [References]
[1] SERGEI I. SCHUKIN Olga V Z Vladymyr G Zinkovsky. Elimination kinetics of the novel prodrug cinazepam possessing psychotropic activity in mice[J]. Pharmacological Reports, 2011, 63 5: Pages 1093-1100. DOI: 10.1016/s1734-1140(11)70628-4 |
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