| Identification | Back Directory | [Name]
BMS 986188 | [CAS]
1776115-10-6 | [Synonyms]
BMS 986188
9-(4-(2-bromobenzyloxy)phenyl)-3,3,6,6-tetramethyl-3,4,5,6,7,9-hexahydro-1H-xanthene-1,8(2H)-dione
1H-Xanthene-1,8(2H)-dione, 9-[4-[(2-bromophenyl)methoxy]phenyl]-3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl- | [Molecular Formula]
C30H31BrO4 | [MDL Number]
MFCD34565177 | [MOL File]
1776115-10-6.mol | [Molecular Weight]
535.47 |
| Chemical Properties | Back Directory | [storage temp. ]
Store at -20°C | [solubility ]
DMF: 1mg/mL; DMF:PBS (pH 7.2) (1:2): 0.3mg/mL; DMSO: slightly soluble; Ethanol: slightly soluble | [form ]
A crystalline solid | [color ]
Off-white to light yellow |
| Hazard Information | Back Directory | [Description]
BMS-986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor. | [Uses]
BMS-986188 is a selective positive allosteric modulator of δ-opioid receptor with an EC50 of 0.05 μM[1]. | [References]
[1] Burford NT, et al. Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptor. J Med Chem. 2015 May 28;58(10):4220-9. DOI:10.1021/acs.jmedchem.5b00007 |
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