| Identification | Back Directory | [Name]
cis MZ 1 | [CAS]
1797406-72-4 | [Synonyms]
cis MZ 1
(2S,4S)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide | [Molecular Formula]
C49H60ClN9O8S2 | [MDL Number]
MFCD30742946 | [MOL File]
1797406-72-4.mol | [Molecular Weight]
1002.64 |
| Hazard Information | Back Directory | [Uses]
cis-MZ 1 is a negative control of MZ 1 (HY-107425). cis-MZ 1 is a PROTAC targeting to BRD4[1]. | [IC 50]
BRD4(BD1BD2) | [storage]
Store at -20°C | [References]
[1] Zengerle M, et al. Selective Small Molecule Induced Degradation of the BET Bromodomain Protein BRD4. ACS Chem Biol. 2015 Aug 21;10(8):1770-7. DOI:10.1021/acschembio.5b00216 |
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