| Identification | Back Directory | [Name]
KDM4D-IN-1 | [CAS]
2098902-68-0 | [Synonyms]
KDM4D-IN-1
KDM4D-IN-10r
KDM4D-IN-1, >98%
KDM4D inhibitor 1
Pyrazolo[1,5-a]pyrido[3,2-e]pyrimidine-3-carbonitrile, 4,5-dihydro-2-methyl-5-oxo- | [Molecular Formula]
C11H7N5O | [MDL Number]
MFCD31544339 | [MOL File]
2098902-68-0.mol | [Molecular Weight]
225.21 |
| Chemical Properties | Back Directory | [Boiling point ]
366.2±42.0 °C(Predicted) | [density ]
1.58±0.1 g/cm3(Predicted) | [storage temp. ]
Store at -20°C | [solubility ]
DMSO : 6 mg/mL (26.64 mM) | [form ]
Solid | [pka]
10.33±0.20(Predicted) | [color ]
Light yellow to khaki |
| Hazard Information | Back Directory | [Uses]
KDM4D-IN-1 is a new histone lysine demethylase 4D (KDM4D) inhibitor with an IC50 value of 0.41±0.03 μM. | [IC 50]
KDM4 | [References]
[1] Fang Z, et al. Discovery of pyrazolo[1,5-a]pyrimidine-3-carbonitrile derivatives as a new class of histone lysine demethylase 4D (KDM4D) inhibitors. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3201-3204. DOI:10.1016/j.bmcl.2017.05.002 |
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| Company Name: |
BOC Sciences
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| Tel: |
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| Website: |
https://www.bocsci.com |
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