| Identification | Back Directory | [Name]
Benzamide, N-[2-[4-(4-chlorophenyl)-1-piperazinyl]ethyl]-3-methoxy- | [CAS]
219125-63-0 | [Synonyms]
Dopamine D4 receptor ligand 2
Benzamide, N-[2-[4-(4-chlorophenyl)-1-piperazinyl]ethyl]-3-methoxy- | [Molecular Formula]
C20H24ClN3O2 | [MOL File]
219125-63-0.mol | [Molecular Weight]
373.88 |
| Hazard Information | Back Directory | [Uses]
Dopamine D4 receptor ligand 2 (compound 17) is a potent and selective dopamine D4 ligand with IC50 values of 0.057, >1000, 220, 270 nM for D4, D2, 5-HT1A, α1, respectively[1]. | [IC 50]
D4 Receptor: 0.057 nM (IC50); D2 Receptor: >1000 nM (IC50); 5-HT1A: 220 nM (IC50); α1: 270 nM (IC50) | [References]
[1] Perrone R, et al. N-[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide: a potent and selective dopamine D4 ligand. J Med Chem. 1998 Nov 19;41(24):4903-9. DOI:10.1021/jm981041x |
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