| Identification | Back Directory | [Name]
fluphenazine O-enantate | [CAS]
2746-81-8 | [Synonyms]
moditen enanthate
fluphenazine O-enantate
Fluphenazine enantate CRS
Fluphenazine Decanoate Impurity 3 (Fluphenazine Decanoate EP Impurity C)
2-[4-[3-[2-(Trifluoromethyl)phenothiazin-10-yl]propyl]-1-piperazinyl]ethyl heptanoate
2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]propyl]piperazin-1-yl]ethyl heptanoate
enanthic acid 2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]propyl]piperazin-1-yl]ethyl ester
Heptanoic acid, 2-4-3-2-(trifluoromethyl)-10H-phenothiazin-10-ylpropyl-1-piperazinylethyl ester | [EINECS(EC#)]
220-385-0 | [Molecular Formula]
C29H38F3N3O2S | [MDL Number]
MFCD00866641 | [MOL File]
2746-81-8.mol | [Molecular Weight]
549.698 |
| Chemical Properties | Back Directory | [Appearance]
Pale yellow, viscous liquid or yellow solid. | [Melting point ]
184.5°C | [Boiling point ]
629.4±55.0 °C(Predicted) | [density ]
1.1661 (estimate) | [storage temp. ]
2-8°C | [solubility ]
Practically insoluble in water, very soluble in ethanol and in methylene chloride, freely soluble in methanol. | [form ]
neat | [pka]
7.32±0.10(Predicted) | [Major Application]
pharmaceutical (small molecule) | [InChIKey]
LRWSFOSWNAQHHW-UHFFFAOYSA-N | [SMILES]
FC(F)(F)c1cc2c(cc1)Sc3c(cccc3)N2CCCN4CCN(CC4)CCOC(=O)CCCCCC |
| Hazard Information | Back Directory | [Chemical Properties]
Pale yellow, viscous liquid or yellow solid. | [Uses]
Antipsychotic. | [Definition]
ChEBI: Fluphenazine enanthate is a member of phenothiazines. | [in vivo]
Fluphenazine enanthate (2,4, 8 mg/kg; IM) significant inhibition of the avoidance performance is observed as long as 16, 23, and 28 days, respectively[1].
Fluphenazine enanthate (8 mg/kg) drinking behavior is almost completely suppressed for 24 hours immediately following the administration[1].
Fluphenazine enanthate (8 mg/kg) produces transient body weight Iosses in the rats[1]. | Animal Model: | Fifty-four male adult rats of Wistar strain[1] | | Dosage: | 2, 4, and 8 mg/kg | | Administration: | Index medicus (IM ) | | Result: | Three doses of Fluphenazine enanthate significant inhibition of the avoidance performance was observed as long as 16, 23, and 28 days, respectively. |
|
| Safety Data | Back Directory | [RIDADR ]
3249 | [WGK Germany ]
WGK 3 | [HazardClass ]
6.1(b) | [PackingGroup ]
III | [Storage Class]
6.1C - Combustible acute toxic Cat.3
toxic compounds or compounds which causing chronic effects | [Hazard Classifications]
Acute Tox. 3 Oral
Repr. 1A |
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BOC Sciences
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16314854226 |
| Website: |
www.bocsci.com |
| Company Name: |
Merck KGaA
|
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21-20338288 |
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www.sigmaaldrich.cn |
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