1-Azetidinesulfonamide(9CI)
- CAS No.
- 654073-32-2
- Chemical Name:
- 1-Azetidinesulfonamide(9CI)
- Synonyms
- 102882;CPD1543-A9;1-Azetidinesulfonamide;azetidine-1-sulfonaMide;azetidine-1-sulphonamide;1-Azetidinesulfonamide(9CI);azetidine-1-sulfonamide - [A87170]
- CBNumber:
- CB01282980
- Molecular Formula:
- C3H8N2O2S
- Molecular Weight:
- 136.17
- MDL Number:
- MFCD18806627
- MOL File:
- 654073-32-2.mol
- MSDS File:
- SDS
| Boiling point | 276.3±23.0 °C(Predicted) |
|---|---|
| Density | 1.51±0.1 g/cm3(Predicted) |
| storage temp. | Sealed in dry,Store in freezer, under -20°C |
| pka | 11.52±0.20(Predicted) |
| Appearance | White to off-white Solid |
| InChI | InChI=1S/C3H8N2O2S/c4-8(6,7)5-2-1-3-5/h1-3H2,(H2,4,6,7) |
| InChIKey | STIUWSWFXIBBKI-UHFFFAOYSA-N |
| SMILES | N1(S(N)(=O)=O)CCC1 |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS07 |
|---|---|
| Signal word | Warning |
| Hazard statements | H335-H319-H315 |
| Precautionary statements | P264-P280-P305+P351+P338-P337+P313P-P264-P280-P302+P352-P321-P332+P313-P362 |
1-Azetidinesulfonamide(9CI) price More Price(31)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Biosynth | EBB07332 | Azetidine-1-sulfonamide | 654073-32-2 | 1g | $318.6 | 2026-06-04 | Buy |
| Biosynth | EBB07332 | Azetidine-1-sulfonamide | 654073-32-2 | 10g | $1534 | 2026-06-04 | Buy |
| Matrix Scientific | 300489 | Azetidine-1-sulfonamide | 654073-32-2 | 100.00mg | $69 | 2026-05-19 | Buy |
| Matrix Scientific | 300489 | Azetidine-1-sulfonamide | 654073-32-2 | 250.00mg | $84 | 2026-05-19 | Buy |
| Matrix Scientific | 300489 | Azetidine-1-sulfonamide | 654073-32-2 | 1.00g | $184 | 2026-05-19 | Buy |
1-Azetidinesulfonamide(9CI) Chemical Properties, Uses, Production
Synthesis
1271835-78-9
654073-32-2
The general procedure for the synthesis of 1-azetidinylsulfonamide using the compound (CAS:1271835-78-9) as starting material was as follows: palladium hydroxide (20%, 350 mg), benzyl (azetidin-1-ylsulfonyl) carbamate (1.49 g, 5.5 mmol), and 1-methyl-1,4-cyclohexadiene (10.7 g, 0.11 mol) of the The mixture was dissolved in methanol (35 mL) and the reaction was stirred at 60 °C under nitrogen protection overnight. After completion of the reaction, the mixture was cooled to room temperature, filtered through a diatomaceous earth pad, and the filtrate was concentrated in vacuum to afford 1-azetidinesulfonamide (437 mg, 58% yield) as a solid product. The product was characterized by 1H NMR (400 MHz, CD3OD) with chemical shifts δ of 2.15 (quintuple peak, 2H) and 3.78 (triplet peak, 4H).The corresponding mass ions were not detected by LCMS analysis.
References
[1] Patent: WO2013/88315, 2013, A1. Location in patent: Page/Page column 75
[2] Patent: WO2013/102826, 2013, A1. Location in patent: Page/Page column 91
1-Azetidinesulfonamide(9CI) Preparation Products And Raw materials
Raw materials
Preparation Products
1-Azetidinesulfonamide(9CI) Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Wuxi Donghe Pharmaceutical Technology Co., Ltd. | 63313187 15358055255 | 63313187@qq.com | China | 1981 | 58 |
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