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amauromine

amauromine structure

CAS No.: 88360-87-6

Chemical Name:: amauromine

Synonyms: WF-6237;FR-900220;amauromine;Antibiotic FR-900220;4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione;4a-bromo-8-methoxy-1,4a,5,10a-tetrahydropyrimido[5,4-b]quinoline-2,4,10(3h)-trione;(5aS,7aS,8aR,13aS,15aS,16aR)-8a,16a-Bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-pyrazino[1'',2'':1,5;(5aS)-8aα,16aα-Bis(1,1-dimethyl-2-propenyl)-5aα,8,8a,13,13aα,15aβ,16,16a-octahydropyrazino[1'',2'':1,5:4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aβH)-dione;4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione, 8a,16a-bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-, (5aS,7aS,8aR,13aS,15aS,16aR)-

CBNumber:: CB11327574

Molecular Formula:: C32H36N4O2

Molecular Weight:: 508.662

MDL Number:: MFCD01939909

MOL File:: 88360-87-6.mol

Last updated:2023-06-30 15:45:59

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amauromine Properties

Boiling point	689.9±55.0 °C(Predicted)
Density	1.28±0.1 g/cm3(Predicted)
storage temp.	Store at -20°C
solubility	DMSO: Soluble; Ethanol: Soluble; Methanol: Soluble
form	A solid
pka	3.26±0.60(Predicted)
color	Brown

SAFETY

Risk and Safety Statements

Symbol(GHS)

GHS07

Signal word

Warning

Hazard statements

H302+H312+H332

Precautionary statements

P261-P264-P270-P271-P280-P301+P312-P302+P352-P304+P340-P321-P330-P362+P364-P501

Toxicity

LD50 intraperitoneal in mouse: > 200mg/kg

NFPA 704

	0
3		0

amauromine price More Price(6)

Manufacturer	Product number	Product description	CAS number	Packaging	Price	Updated	Buy
Cayman Chemical	23886	Amauromine ≥98%	88360-87-6	250μg	$79	2024-03-01	Buy
Cayman Chemical	23886	Amauromine ≥98%	88360-87-6	1mg	$219	2024-03-01	Buy
Usbiological	044497	Amauromine	88360-87-6	250ug	$290	2021-12-16	Buy
TRC	A575993	Amauromine	88360-87-6	2.5mg	$295	2021-12-16	Buy
American Custom Chemicals Corporation	INB0003887	AMAUROMINE 95.00%	88360-87-6	5MG	$501.22	2021-12-16	Buy

Product number	Packaging	Price	Buy
23886	250μg	$79	Buy
23886	1mg	$219	Buy
044497	250ug	$290	Buy
A575993	2.5mg	$295	Buy
INB0003887	5MG	$501.22	Buy

amauromine Chemical Properties,Uses,Production

Description

Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB₁ that is selective for CB₁ (K_i = 178 nM; K_b = 66.6 nM) over CB₂, with no activity at CB₂ receptors at concentrations up to 10 μM. It is also an antagonist of GPR18 (IC₅₀ = 3.74 μM). Amauromine has vasodilatory activity.

Uses

Amauromine is a CB1 and Calcium Channel antagonist.

storage

+4°C

amauromine synthesis

Synthesis of amauromine from L-Tryptophan, N,1-bis[(1,1-dimethylethoxy)carbonyl]-, methyl ester

amauromine Preparation Products And Raw materials

Raw materials

L-Tryptophan, N,1-bis[(1,1-dimethylethoxy)carbonyl]-, methyl ester

Preparation Products

amauromine Suppliers

Global( 24)Suppliers

Supplier	Tel	Email	Country	ProdList	Advantage
Hangzhou MolCore BioPharmatech Co.,Ltd.	+86-057181025280; +8617767106207	sales@molcore.com	China	49739	58
Shanghai EFE Biological Technology Co., Ltd.	021-65675885 18964387627	info@efebio.com	China	9709	58
Shanghai Hongye Biotechnology Co. Ltd	400-9205774	sales@glpbio.cn	China	6870	58
Meng Cheng Technology (Shanghai) Co., LTD	400-820-6829	sales@mitachieve.com	China	8864	58
Energy Chemical	021-58432009 400-005-6266	marketing@energy-chemical.com	China	44941	58
TargetMol Chemicals Inc.	4008200310	marketing@tsbiochem.com	China	24017	58

Supplier	Advantage
Hangzhou MolCore BioPharmatech Co.,Ltd.	58
Shanghai EFE Biological Technology Co., Ltd.	58
Shanghai Hongye Biotechnology Co. Ltd	58
Meng Cheng Technology (Shanghai) Co., LTD	58
Energy Chemical	58
TargetMol Chemicals Inc.	58

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amauromine (5aS)-8aα,16aα-Bis(1,1-dimethyl-2-propenyl)-5aα,8,8a,13,13aα,15aβ,16,16a-octahydropyrazino[1'',2'':1,5:4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aβH)-dione Antibiotic FR-900220 FR-900220 WF-6237 (5aS,7aS,8aR,13aS,15aS,16aR)-8a,16a-Bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-pyrazino[1'',2'':1,5 4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione 4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione, 8a,16a-bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-, (5aS,7aS,8aR,13aS,15aS,16aR)- 4a-bromo-8-methoxy-1,4a,5,10a-tetrahydropyrimido[5,4-b]quinoline-2,4,10(3h)-trione 88360-87-6 C32H36N4O2