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ChemicalBook >> CAS DataBase List >>(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Structure
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 structure
CAS No.
208706-12-1
Chemical Name:
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
Synonyms
264;3'R/1R;3'S)-L-054;(1R,1’S)-DuanPhos;S)-L-054,264;-iodo-1’(1R,1S,3R/1R,1R,3'S);S)-Octahydro-1-(2’-Hydroxy pravastatin sodium salt
CBNumber:
CB52453421
Molecular Formula:
C33H41N5O2
Molecular Weight:
539.71
MDL Number:
MFCD09971077
MOL File:
208706-12-1.mol
Last updated:2023-06-30 15:45:59
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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Properties

Boiling point 865.2±65.0 °C(Predicted)
Density 1.25±0.1 g/cm3(Predicted)
storage temp. Store at +4°C
solubility Soluble to 50 mM in DMSO and to 100 mM in ethanol
form Powder
pka 12.79±0.20(Predicted)

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 price More Price(6)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Tocris 2444 (1R,1S,3R/1R,1R,3'S)-L-054,264 ≥96%(HPLC) 208706-12-1 10 $289 2021-12-16 Buy
Tocris 2444 (1R,1S,3R/1R,1R,3'S)-L-054,264 ≥96%(HPLC) 208706-12-1 1 $134 2021-12-16 Buy
TRC A633290 N-​[(1R)​-​2-​[[[3-​(Aminomethyl)​cyclohexyl]​methyl]​amino]​-​1-​(1H-​indol-​3-​ylmethyl)​-​2-​oxoethyl]​-spiro[1H-​indene-​1,​4''-​piperidine]​-​1''-​carboxamide 208706-12-1 2.5mg $315 2021-12-16 Buy
ApexBio Technology B7057 (1R,1'S,3'R/1R,1'R,3'S)-L-054,264 208706-12-1 10mg $423 2021-12-16 Buy
American Custom Chemicals Corporation API0009813 (1R,1'S,3'R/1R,1'R,3'S)-L-054,264 95.00% 208706-12-1 5MG $504.41 2021-12-16 Buy
Product number Packaging Price Buy
2444 10 $289 Buy
2444 1 $134 Buy
A633290 2.5mg $315 Buy
B7057 10mg $423 Buy
API0009813 5MG $504.41 Buy

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Chemical Properties,Uses,Production

Uses

Somatostatin receptors are often overexpressed in tumours and are potential therapeutic targets. Somatostatin receptor agonists can be used to study signaling pathways related somatostatin receptor.N-?[(1R)?-?2-?[[[3-?(Aminomethyl)?cyclohexyl]?methyl]?amino]?-?1-?(1H-?indol-?3-?ylmethyl)?-?2-?oxoethyl]?-spiro[1H-?indene-?1,?4''-?piperidine]?-?1''-?carboxamide is a selective somatostatin sst2 receptor agonist.

Biological Activity

Potent and selective somatostatin sst 2 receptor agonist (K i values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst 2 , sst 1 , sst 4 , sst 3 and sst 5 receptors respectively).

storage

Store at +4°C

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Preparation Products And Raw materials

Raw materials

Preparation Products

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Suppliers

Global( 15)Suppliers
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TargetMol Chemicals Inc. 		+1-781-999-5354 +1-00000000000 marketing@targetmol.com United States 19892 58
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Aladdin Scientific 		+1-833-552-7181 sales@aladdinsci.com United States 52927 58
3B Pharmachem (Wuhan) International Co.,Ltd. 821-50328103-801 18930552037 3bsc@sina.com China 15848 69
Shanghai T&W Pharmaceutical Co., Ltd. +86 21 61551611 China 9901 58
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Shanghai Universal Biotech Co.,Ltd 18768175414 gaojun@univ-bio.com China 24998 58
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Henan Alpha Chemical Co., Ltd. 0371-55013243 15324716602 2853979810@qq.com China 9623 58
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TargetMol Chemicals Inc. 		58
Hangzhou MolCore BioPharmatech Co.,Ltd. 		58
Aladdin Scientific 		58
3B Pharmachem (Wuhan) International Co.,Ltd. 69
Shanghai T&W Pharmaceutical Co., Ltd. 58
EMMX Biotechnology LLC 60
BOC Sciences 65
Shanghai Universal Biotech Co.,Ltd 58
TargetMol Chemicals Inc. 58
Henan Alpha Chemical Co., Ltd. 58

208706-12-1((1R,1'S,3'R/1R,1'R,3'S)-L-054,264)Related Search:

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 SPIRO[INDENE-1,4'-PIPERIDINE] 1,3-Cyclohexanebis(methylamine)
N-[(1R)-2-[[[(1S*,3R*)-3-(AMINOMETHYL)CYCLOHEXYL]METHYL]AMINO]-1-(1H-INDOL-3-YLMETHYL)-2-OXOETHYL]SPIRO[1H-INDENE-1,4'-PIPERIDINE]-1'-CARBOXAMIDE S)-L-054,264 (1R,1'S,3'R/1R,1'R,3'S)-L-054,264 -methylethyl)-7a-methyl-inden-4-one S)-DuanPhos -Hydroxy pravastatin sodium salt (1R,1&rsquo -iodo-1&rsquo S)-Octahydro-1-(2&rsquo -methylethyl)-7a-methyl-inden-4-ol -(((2-Aminopropane-1,3-diyl)bis(oxy))bis(methylene))bis(phenylcyclopropanecarboxamide) Spiro[1H-indene-1,4'-piperidine]-1'-carboxamide, N-[(1R)-2-[[[3-(aminomethyl)cyclohexyl]methyl]amino]-1-(1H-indol-3-ylmethyl)-2-oxoethyl]- N-?[(1R)?-?2-?[[[3-?(Aminomethyl)?cyclohexyl]?methyl]?amino]?-?1-?(1H-?indol-?3-?ylmethyl)?-?2-?oxoethyl]?-spiro[1H-?indene-?1,?4'-?piperidine]?-?1'-?carboxamide (1R,1S,3R/1R,1R,3'S) 264 3'R/1R 3'S)-L-054 (1R,1'S,3'R/1R,1'R,3'S)L054,264,(1R,1'S,3'R/1R,1'R,3'S) L 054,264 N-((2R)-1-(((3-(Aminomethyl)cyclohexyl)methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide (1R,1'S,3'R/1R,1'R,3'S)-L-054,264 208706-12-1 C33H41N5O2