RO-31-7549 化学特性,用途語,生産方法
使用
It is a potent inhibitor of protein kinase C (PKC) activity.
一般的な説明
A cell permeable, reversible, selective protein kinase C (PKC) inhibitor (IC
50 = 158 nM for rat brain PKC) that acts at the ATP binding site of PKC. Does not inhibit the tyrosine phosphorylation or the activation of phospholipase Cγ
1. Exhibits some degree of PKC isozyme specificity (IC
50 = 53 nM for PKC
α, 195 nM for PKC
βI, 163 nM for PKC
βII, 213 nM for PKC
γ, and 175 nM for PKC
ε). Inhibits carbachol-evoked noradrenaline release (IC
50 = 600 nM).
Biochem/physiol Actions
Cell permeable: yes
RO-31-7549 上流と下流の製品情報
原材料
準備製品