セファセトリル 化学特性,用途語,生産方法
効能
抗生物質, 細胞壁合成阻害薬
化学的特性
Pale Beige Solid
抗菌性
Its spectrum resembles that of cefalotin. Following an intramuscular
dose of 1 g, a peak plasma concentration around
15 mg/L is achieved at 1 h. About 25% is bound to plasma protein. Penetration into the CSF is limited. About 80% of
the drug is excreted in the urine, producing concentrations
in excess of 1 g/L, 25% of which is in the desacetylated form.
Clearance is depressed by probenecid and in renal failure.
Little is excreted in the bile.
Manifestations of hypersensitivity in patients not known
to be allergic to β-lactam antibiotics are common. It is no
longer used.
セファセトリル 上流と下流の製品情報
原材料
準備製品