GR113808

GR113808 価格 もっと(4)

メーカー	製品番号	製品説明	CAS番号	包装	価格	更新時間	購入
富士フイルム和光純薬株式会社(wako)	W01TOC1322	GR113808 GR 113808	144625-51-4	10mg	￥68000	2024-03-01	購入
富士フイルム和光純薬株式会社(wako)	W01TOC1322	GR113808 GR 113808	144625-51-4	50mg	￥288000	2024-03-01	購入
Sigma-Aldrich Japan	G5918	≥98% (HPLC), solid GR 113808 ≥98% (HPLC), solid	144625-51-4	10mg	￥39300	2024-03-01	購入
Sigma-Aldrich Japan	G5918	≥98% (HPLC), solid GR 113808 ≥98% (HPLC), solid	144625-51-4	50mg	￥131000	2024-03-01	購入

GR113808 化学特性,用途語,生産方法

使用

GR 113808 has been used as a serotonin receptor 4 (5-HT4R) blocker to study its effects on the calcium (Ca²⁺) transients in rat ventricular cardiomyocytes. It has also been used as a 5-HT4R antagonist to study its effects on de novo enteric neurogenesis in post-embryonic zebrafish.

定義

ChEBI: An indolyl carboxylate ester obtained by formal condensation between the carboxy group of 1-methylindole-3-carboxylic acid with the hydroxy group of N-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}methanesulfonamide.

生物活性

Potent, selective 5-HT 4 receptor antagonist (pK B = 9.43 in human colonic muscle, and K d = 0.15 nM for binding to cloned human 5-HT 4 receptors). Displays > 300-fold selectivity over 5-HT 1A , 5-HT 1B , 5-HT 2A , 5-HT 2C and 5-HT 3 receptors.

GR113808 上流と下流の製品情報

原材料

準備製品

GR113808 生産企業

名前	電話番号	電子メール	国籍	製品カタログ	優位度
TargetMol Chemicals Inc.	+1-781-999-5354 +1-00000000000	marketing@targetmol.com	United States	19892	58
Career Henan Chemica Co	+86-0371-86658258 15093356674;	laboratory@coreychem.com	China	30255	58
Aladdin Scientific	+1-833-552-7181	sales@aladdinsci.com	United States	52927	58
3B Pharmachem (Wuhan) International Co.,Ltd.	821-50328103-801 18930552037	3bsc@sina.com	China	15848	69
BOC Sciences	1-631-485-4226; 16314854226	info@bocsci.com	United States	14059	65
Sigma-Aldrich	021-61415566 800-8193336	orderCN@merckgroup.com	China	51471	80
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8449	60
DC Chemicals	021-58447131 13564518121	sales@dcchemicals.com	China	9414	58
ChemeGen(Shanghai) Biotechnology Co.,Ltd.	18818260767	sales@chemegen.com	China	11289	58
Energy Chemical	021-58432009 400-005-6266	marketing1@energy-chemical.com	China	44894	58

144625-51-4(GR113808)キーワード:

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• 144625-51-4
• 1-METHYL-1H-INDOLE-3-CARBOXYLIC ACID, [1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]METHYL ESTER
• 1-[2-(METHYLSULFONYL)-AMINO]ETHYL-4-PIPERIDINYLMETHYL 1-METHYL-1H-INDOLE-3-CARBOXYLATE
• GR 113808;1-METHYL-1H-INDOLE-3-CARBOXYLIC ACID, [1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]METHYL ESTER;1-[2-(METHYLSULFONYL)-AMINO]ETHYL-4-PIPERIDINYLMETHYL 1-METHYL-1H-INDOLE-3-CARBOXYLATE;GR 113808
• 1-Methyl-1H-indole-3-carboxylicacid,[1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]methyles
• GR 113808
• 1H-Indole-3-carboxylic acid, 1-methyl-, [1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]methyl ester
• GR113808
• 1-メチル-1H-インドール-3-カルボン酸[1-[2-[(メチルスルホニル)アミノ]エチル]-4-ピペリジニル]メチル
• 1-メチル-1H-インドール-3-カルボン酸1-[2-(メチルスルホニルアミノ)エチル]ピペリジン-4-イルメチル
• GR-113808
• [1-(2-メタンスルホンアミドエチル)ピペリジン-4-イル]メチル 1-メチル-1H-インドール-3-カルボキシラート
• 1-メチル-1H-インドール-3-カルボン酸1-[2-(メチルスルホニルアミノ)エチル]-4-ピペリジニルメチル