Apalutamide
|
- $14 - $3142
- Product name: Apalutamide
- CAS: 956104-40-8
- MF: C21H15F4N5O2S
- MW: 477.43
- EINECS:807-449-9
- MDL Number:MFCD22380626
- Synonyms:AR509;AR509 100G;ARV-509;ARN-509;ARN 509; ARN509;4-(7-(4-Cyano-3-(trifluoromethyl)phenyl)-8-hydroxy-6-thioxo-5,7-diazaspiro[3.4]octan-5-yl)-2-f;AR509/AR-509;ARN;ARN 509; ARN-509
68 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Axon Medchem
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- Chemenu
- ChemScene
- Crysdot
- DC Chemicals
- Matrix Scientific
- TRC
Package
- 10mM(in 1mL DMSO)
- 1MG
- 10mg
- 25mg
- 10mM*1mLinDMSO(Solution)
- 5MG
- 10mM(in1mLDMSO)
- 10mM*1mLinDMSO(Solid+Solvent)
- 50mg
- 100mg
- 200mg
- 250mg
- 500mg
- 1.00g
- 1g
- 5.00g
- 5g
- 25g
- 25.00g
- Manufactureraablocks
- Product numberAA00IJ5V
- Product description4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 95%
- Packaging25mg
- Price$14
- Updated2026-05-29
- Buy
- Manufactureraablocks
- Product numberAA00IJ5V
- Product description4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98%
- Packaging100mg
- Price$15
- Updated2026-05-29
- Buy
- Manufactureraablocks
- Product numberAA00IJ5V
- Product description4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98%
- Packaging250mg
- Price$25
- Updated2026-05-29
- Buy
- Manufactureraablocks
- Product numberAA00IJ5V
- Product description4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98%
- Packaging1g
- Price$60
- Updated2026-05-29
- Buy
- Manufactureraablocks
- Product numberAA00IJ5V
- Product description4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98%
- Packaging5g
- Price$234
- Updated2026-05-29
- Buy
- Manufactureraablocks
- Product numberAA00IJ5V
- Product description4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98%
- Packaging25g
- Price$988
- Updated2026-05-29
- Buy
- ManufacturerACHEMBLOCK
- Product numberR16071
- Product descriptionARN-509 98%
- Packaging100MG
- Price$45
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberR16071
- Product descriptionARN-509 98%
- Packaging1G
- Price$100
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberR16071
- Product descriptionARN-509 98%
- Packaging5G
- Price$290
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberY0375
- Product descriptionBenzamide,4-[7-[6-cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methyl-
- Packaging1g
- Price$1987
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0015790
- Product descriptionARN-509 95.00%
- Packaging1MG
- Price$148.05
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0015790
- Product descriptionARN-509 95.00%
- Packaging5MG
- Price$500.82
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8364
- Product descriptionARN-509
- Packaging10mM(in 1mL DMSO)
- Price$105
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8364
- Product descriptionARN-509
- Packaging10mg
- Price$110
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberA8364
- Product descriptionARN-509
- Packaging5mg
- Price$64
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberA8364
- Product descriptionARN-509
- Packaging10mM(in1mLDMSO)
- Price$77
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA00IJ5V | 4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 95% | 25mg | $14 | 2026-05-29 | Buy |
| aablocks | AA00IJ5V | 4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98% | 100mg | $15 | 2026-05-29 | Buy |
| aablocks | AA00IJ5V | 4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98% | 250mg | $25 | 2026-05-29 | Buy |
| aablocks | AA00IJ5V | 4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98% | 1g | $60 | 2026-05-29 | Buy |
| aablocks | AA00IJ5V | 4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98% | 5g | $234 | 2026-05-29 | Buy |
| aablocks | AA00IJ5V | 4-[7-[6-Cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methylbenzamide 98% | 25g | $988 | 2026-05-29 | Buy |
| ACHEMBLOCK | R16071 | ARN-509 98% | 100MG | $45 | 2026-05-27 | Buy |
| ACHEMBLOCK | R16071 | ARN-509 98% | 1G | $100 | 2026-05-27 | Buy |
| ACHEMBLOCK | R16071 | ARN-509 98% | 5G | $290 | 2026-05-27 | Buy |
| AK Scientific | Y0375 | Benzamide,4-[7-[6-cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methyl- | 1g | $1987 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0015790 | ARN-509 95.00% | 1MG | $148.05 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0015790 | ARN-509 95.00% | 5MG | $500.82 | 2021-12-16 | Buy |
| ApexBio Technology | A8364 | ARN-509 | 10mM(in 1mL DMSO) | $105 | 2021-12-16 | Buy |
| ApexBio Technology | A8364 | ARN-509 | 10mg | $110 | 2026-05-06 | Buy |
| ApexBio Technology | A8364 | ARN-509 | 5mg | $64 | 2026-05-06 | Buy |
| ApexBio Technology | A8364 | ARN-509 | 10mM(in1mLDMSO) | $77 | 2026-05-06 | Buy |
Properties
Density :1.59±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :≥23.85 mg/mL in DMSO; insoluble in H2O; ≥7.33 mg/mL in EtOH
form :solid
pka :13.83±0.46(Predicted)
color :White to off-white
InChI :InChI=1S/C21H15F4N5O2S/c1-27-17(31)13-4-3-11(8-15(13)22)30-19(33)29(18(32)20(30)5-2-6-20)12-7-14(21(23,24)25)16(9-26)28-10-12/h3-4,7-8,10H,2,5-6H2,1H3,(H,27,31)
InChIKey :HJBWBFZLDZWPHF-UHFFFAOYSA-N
SMILES :C(NC)(=O)C1=CC=C(N2C(=S)N(C3=CC(C(F)(F)F)=C(C#N)N=C3)C(=O)C32CCC3)C=C1F
storage temp. :Store at -20°C
solubility :≥23.85 mg/mL in DMSO; insoluble in H2O; ≥7.33 mg/mL in EtOH
form :solid
pka :13.83±0.46(Predicted)
color :White to off-white
InChI :InChI=1S/C21H15F4N5O2S/c1-27-17(31)13-4-3-11(8-15(13)22)30-19(33)29(18(32)20(30)5-2-6-20)12-7-14(21(23,24)25)16(9-26)28-10-12/h3-4,7-8,10H,2,5-6H2,1H3,(H,27,31)
InChIKey :HJBWBFZLDZWPHF-UHFFFAOYSA-N
SMILES :C(NC)(=O)C1=CC=C(N2C(=S)N(C3=CC(C(F)(F)F)=C(C#N)N=C3)C(=O)C32CCC3)C=C1F
Safety Information
| Symbol(GHS): |
|
||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Signal word: | Warning | ||||||||||||||
| Hazard statements: |
|
||||||||||||||
| Precautionary statements: |
|
Description
ARN-509 is a selective and competitive androgen receptor inhibitor with IC50 of 16 nM in a cell-free assay, useful for prostate cancer treatment. Phase 3.More related product prices
Olaparib Ibrutinib Galeterone Bicalutamide 749927-69-3 3-nitro-4-((tetrahydro-2H-pyran-4-yl)MethylaMino)benzenesulfonaMide abt199 int 2 1-((4'-chloro-5,5-dimethyl-3,4,5,6-tetrahydro-[1,1'-biphenyl]-2-yl)methyl)piperazine dihydrochloride ABT-199 tert-butyl 2-((1H-pyrrolo[2,3-b]pyridin-5-yl)oxy)-4-bromobenzoate Y27632 (hydrochloride) Enzalutamide (MDV3100)Related product price
-
Olaparib
$11-2994.75 -
Ibrutinib
$5-1360 -
Galeterone
$28-2650
Suppliers and manufacturers
Chongqing Chemieliva Pharmaceutical Co., Ltd.
Changzhou Yongfeng Biomedicine Co. Ltd.
Hangzhou Xinbaisi Biomedical Co., Ltd.
Junyu Chemexpress Co., Ltd.
Zhengzhou Runkai Pharmaceutical Technology Co., Ltd
Beijing Hope Pharmaceutical Co., Ltd.
CHENGHUI PHARMACEUTICAL GROUP LTD
Shanghai Famo Biotechnology Co., Ltd.
Shanghai Boyle Chemical Co., Ltd.
ChemFuture PharmaTech (Jiangsu) Ltd