BAY-876
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- $32 - $4741
- Product name: BAY-876
- CAS: 1799753-84-6
- MF: C24H16F4N6O2
- MW: 496.42
- EINECS:
- MDL Number:MFCD30377201
- Synonyms:N4-[1-[(4-cyanophenyl)methyl]-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]-7-fluoro-2,4-Quinolinedicarboxamide;BAY-876;N4-(1-(4-cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide;CS-2442;BAY876;BAY 876;BAY-876 >=98% (HPLC);2,4-Quinolinedicarboxamide, N4-[1-[(4-cyanophenyl)methyl]-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]-7-fluoro-;Inhibitor,metabolism,transporter,ovarian,BAY876,BAY 876,glycolytic,cancer,Glucose transporter,glucose,inhibit,BAY-876,orally,GLUT
66 prices
Selected condition:
Brand
- aablocks
- AK Scientific
- Ambeed
- American Custom Chemicals Corporation
- Arctom
- Axon Medchem
- Biosynth
- Cayman Chemical
- Chemenu
- ChemScene
- Crysdot
- DC Chemicals
- Sigma-Aldrich
- Tocris
- TRC
Package
- 5mg
- 5
- 2mg
- 25
- 1mg
- 10mM*1mLinDMSO(Solid+Solvent)
- 10mM*1mLinDMSO
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- 1000mg
- 500mg
- 10mM*1mLinDMSO(Solution)
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98%
- Packaging10mg
- Price$105
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98
- Packaging25mg
- Price$217
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98
- Packaging50mg
- Price$317
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98%
- Packaging100mg
- Price$418
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98%
- Packaging5mg
- Price$70
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98%
- Packaging2mg
- Price$46
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98%
- Packaging1mg
- Price$32
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98%
- Packaging250mg
- Price$829
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0021GO
- Product descriptionBAY-876 98%
- Packaging1g
- Price$2075
- Updated2026-05-28
- Buy
- ManufacturerAK Scientific
- Product number2583EF
- Product description4-N-[1-[(4-Cyanophenyl)methyl]-5-methyl-3-(trifluoromethyl)pyrazol-4-yl]-7-fluoroquinoline-2,4-dicarboxamide
- Packaging10mg
- Price$259
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA863389
- Product descriptionN4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+%
- Packaging100mg
- Price$312
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA863389
- Product descriptionN4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+%
- Packaging50mg
- Price$240
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA863389
- Product descriptionN4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+%
- Packaging2mg
- Price$63
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA863389
- Product descriptionN4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+%
- Packaging5mg
- Price$82
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA863389
- Product descriptionN4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+%
- Packaging10mg
- Price$122
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA863389
- Product descriptionN4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+%
- Packaging1g
- Price$1549
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA0021GO | BAY-876 98% | 10mg | $105 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98 | 25mg | $217 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98 | 50mg | $317 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98% | 100mg | $418 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98% | 5mg | $70 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98% | 2mg | $46 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98% | 1mg | $32 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98% | 250mg | $829 | 2026-05-28 | Buy |
| aablocks | AA0021GO | BAY-876 98% | 1g | $2075 | 2026-05-28 | Buy |
| AK Scientific | 2583EF | 4-N-[1-[(4-Cyanophenyl)methyl]-5-methyl-3-(trifluoromethyl)pyrazol-4-yl]-7-fluoroquinoline-2,4-dicarboxamide | 10mg | $259 | 2021-12-16 | Buy |
| Ambeed | A863389 | N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+% | 100mg | $312 | 2021-12-16 | Buy |
| Ambeed | A863389 | N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+% | 50mg | $240 | 2021-12-16 | Buy |
| Ambeed | A863389 | N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+% | 2mg | $63 | 2021-12-16 | Buy |
| Ambeed | A863389 | N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+% | 5mg | $82 | 2021-12-16 | Buy |
| Ambeed | A863389 | N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+% | 10mg | $122 | 2021-12-16 | Buy |
| Ambeed | A863389 | N4-(1-(4-Cyanobenzyl)-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)-7-fluoroquinoline-2,4-dicarboxamide 99+% | 1g | $1549 | 2021-12-16 | Buy |
Properties
Melting point :>250oC (dec.)
Boiling point :632.3±55.0 °C(Predicted)
Density :1.48±0.1 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO (Slightly), Methanol (Slightly)
form :powder
pka :10.33±0.70(Predicted)
color :white to beige
InChIKey :BKLJDIJJOOQUFG-UHFFFAOYSA-N
SMILES :FC1=CC=C2C(N=C(C(N)=O)C=C2C(NC3=C(C)N(CC4=CC=C(C#N)C=C4)N=C3C(F)(F)F)=O)=C1
Boiling point :632.3±55.0 °C(Predicted)
Density :1.48±0.1 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO (Slightly), Methanol (Slightly)
form :powder
pka :10.33±0.70(Predicted)
color :white to beige
InChIKey :BKLJDIJJOOQUFG-UHFFFAOYSA-N
SMILES :FC1=CC=C2C(N=C(C(N)=O)C=C2C(NC3=C(C)N(CC4=CC=C(C#N)C=C4)N=C3C(F)(F)F)=O)=C1
Safety Information
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Description
BAY-876 is a potent, highly selective, cell-permeable inhibitor of glucose transporter GLUT1. It had an IC50 value of 2 nM in vitro and inhibited glucose uptake by Hela-MaTu cells with an IC50 value of 3.2 nM. BAY-876 was at least 130-fold selective for GLUT1 relative to GLUT2, GLUT3, GLUT4 and a panel of 18 kinases and 68 proteins.BAY-588 is used as a negative control and is available from Sigma.Suppliers and manufacturers
Beijing HwrkChemical Technology Co., Ltd
Dalian Meilun Biotech Co., Ltd.
Haoyuan Chemexpress Co., Ltd.
Bide Pharmatech Ltd.
Shanghai Macklin Biochemical Co.,Ltd.
Sigma-Aldrich
Shanghai Lollane Biological Technology Co.,Ltd.
Shanghaizehan biopharma technology co., Ltd.
Shanghai EFE Biological Technology Co., Ltd.
Shanghai YuanYe Biotechnology Co., Ltd.




