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ChemicalBook >> CAS DataBase List >> Bilastine

Bilastine

Bilastine price.
  • $6 - $2310
  • Product name: Bilastine
  • CAS: 202189-78-4
  • MF: C28H37N3O3
  • MW: 463.62
  • EINECS:
  • MDL Number:MFCD09837814
  • Synonyms:4-[2-[4-[1-(2-Ethoxyethyl)-1H-benziMidazol-2-yl]-1-piperidinyl]ethyl]-α,α-diMethylbenzeneacetic Acid;Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benziMidazol-2-yl]-1-piperidinyl]ethyl]-a,a-diMethyl-;BENZENEACETIC ACID, 4-(2-(4-(1-(2-ETHOXYETHYL)-1H-BENZIMIDAZOL-2-YL)-1-PIPERIDINYL)ETHYL-ALPHA, ALPHA-DIMETHYL-;2-[4-[2-[4-[1-(2-ethoxyethyl)benzoimidazol-2-yl]-1-piperidyl]ethyl]phenyl]-2-methyl-propanoic acid;4-[2-[4-[1-(2-Ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-alpha,alpha-dimethylbenzeneacetic acid;Bilasten;2-[4-[2-[4-[1-(2-ethoxyethyl)benzimidazol-2-yl]piperidin-1-yl]ethyl]phenyl]-2-methylpropanoic acid;the impurity of Bilastine
Price59 Properties Safety Information Description
59 prices
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  • aablocks
  • ACHEMBLOCK
  • AK Scientific
  • Ambeed
  • American Custom Chemicals Corporation
  • ApexBio Technology
  • Arctom
  • Axon Medchem
  • Biosynth
  • Cayman Chemical
  • Chem-Impex
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  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging1mg
  • Price$9
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging10mg
  • Price$15
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging50mg
  • Price$21
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging5mg
  • Price$12
  • Updated2026-05-28
  • Buy
  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging100mg
  • Price$32
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging250mg
  • Price$48
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging1g
  • Price$107
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00281C
  • Product descriptionBenzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98%
  • Packaging5g
  • Price$332
  • Updated2026-05-28
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  • ManufacturerACHEMBLOCK
  • Product number10295
  • Product descriptionBilastine 98%
  • Packaging5G
  • Price$420
  • Updated2026-05-27
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  • ManufacturerACHEMBLOCK
  • Product number10295
  • Product descriptionBilastine 98%
  • Packaging1G
  • Price$135
  • Updated2026-05-27
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  • ManufacturerACHEMBLOCK
  • Product number10295
  • Product descriptionBilastine 98%
  • Packaging100MG
  • Price$45
  • Updated2026-05-27
  • Buy
  • ManufacturerAK Scientific
  • Product number3489AH
  • Product descriptionBilastine
  • Packaging100mg
  • Price$270
  • Updated2021-12-16
  • Buy
  • ManufacturerAmbeed
  • Product numberA325945
  • Product description2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+%
  • Packaging5mg
  • Price$10
  • Updated2021-12-16
  • Buy
  • ManufacturerAmbeed
  • Product numberA325945
  • Product description2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+%
  • Packaging100mg
  • Price$36
  • Updated2021-12-16
  • Buy
  • ManufacturerAmbeed
  • Product numberA325945
  • Product description2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+%
  • Packaging10mg
  • Price$13
  • Updated2021-12-16
  • Buy
  • ManufacturerAmbeed
  • Product numberA325945
  • Product description2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+%
  • Packaging50mg
  • Price$22
  • Updated2021-12-16
  • Buy
Manufacturer Product number Product description Packaging Price Updated Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 1mg $9 2026-05-28 Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 10mg $15 2026-05-28 Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 50mg $21 2026-05-28 Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 5mg $12 2026-05-28 Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 100mg $32 2026-05-28 Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 250mg $48 2026-05-28 Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 1g $107 2026-05-28 Buy
aablocks AA00281C Benzeneacetic acid,4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-α,α-dimethyl- 98% 5g $332 2026-05-28 Buy
ACHEMBLOCK 10295 Bilastine 98% 5G $420 2026-05-27 Buy
ACHEMBLOCK 10295 Bilastine 98% 1G $135 2026-05-27 Buy
ACHEMBLOCK 10295 Bilastine 98% 100MG $45 2026-05-27 Buy
AK Scientific 3489AH Bilastine 100mg $270 2021-12-16 Buy
Ambeed A325945 2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+% 5mg $10 2021-12-16 Buy
Ambeed A325945 2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+% 100mg $36 2021-12-16 Buy
Ambeed A325945 2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+% 10mg $13 2021-12-16 Buy
Ambeed A325945 2-(4-(2-(4-(1-(2-Ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoicacid 98+% 50mg $22 2021-12-16 Buy
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Properties

Melting point :202 °C
Boiling point :639.1±55.0 °C(Predicted)
Density :1.16±0.1 g/cm3(Predicted)
storage temp. :Sealed in dry,Room Temperature
Water Solubility :Insoluble in water
solubility :DMSO:49.3(Max Conc. mg/mL);106.34(Max Conc. mM)
pka :4.40±0.10(Predicted)
form :powder to crystal
color :White to Light yellow
optical activity :-0.2797°(C=0.7419g/100mI, CHCL3, 20°C, 589nm)
InChI :1S/C28H37N3O3/c1-4-34-20-19-31-25-8-6-5-7-24(25)29-26(31)22-14-17-30(18-15-22)16-13-21-9-11-23(12-10-21)28(2,3)27(32)33/h5-12,22H,4,13-20H2,1-3H3,(H,32,33)
InChIKey :ACCMWZWAEFYUGZ-UHFFFAOYSA-N
SMILES :C(N1C2=CC=CC=C2N=C1C1CCN(CCC2C=CC(C(C)(C)C(=O)O)=CC=2)CC1)COCC

Safety Information

Symbol(GHS): Exclamation Mark (GHS07)
Signal word: Warning
Hazard statements:
Code Hazard statements Hazard class Category Signal word Pictogram P-Codes
H302 Harmful if swallowed Acute toxicity,oral Category 4 Warning P264, P270, P301+P312, P330, P501
Precautionary statements:
P280 Wear protective gloves/protective clothing/eye protection/face protection.
P305+P351+P338 IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

Description

Bilastine, a potent and selective histamine H1 receptor antagonist, was approved in Europe in 2010 for the treatment of allergic rhinoconjunctivitis (AR) and urticaria (hives or skin rash). The original synthesis of bilastine involves alkylation of 2-piperidinyl-1H-benzimidazole with a phenethyltosylate, the para position of which is substituted with a dimethyloxazoline moiety serving as a masked carboxylic acid group. Alkylation of the benzimidazole nitrogen with 2-chloroethyl ethyl ether followed by unmasking of the oxazoline moiety with sulfuric acid provided bilastine.
In two major clinical trials, bilastine was effective at relieving allergic rhinitis as assessed by measuring the severity of nasal (obstruction, rhinorrhea, itching, sneezing) and nonnasal (ocular itching, tearing, ocular redness, itching of ears, and/or palate) symptoms.

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Suppliers and manufacturers

Shanghai Boc Chemical Co.,Ltd Shanghai jing Hao pharmaceutical technology co., LTD Tianjin Being Technology Co., Ltd. Shandong Mingfeng Pharmaceutical and Technology Co. Ltd CHENGHUI PHARMACEUTICAL GROUP LTD BOYAN PHARMA Shan Dong FengJin Pharmaceutical Co.,Ltd. BJBXSW Shanghai Boyle Chemical Co., Ltd. J & K SCIENTIFIC LTD.