GSK6853
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- $24 - $2300
- Product name: GSK6853
- CAS: 1910124-24-1
- MF: C22H27N5O3
- MW: 409.48
- EINECS:-0
- MDL Number:MFCD30489734
- Synonyms:GSK6853;GSK6853 >=98% (HPLC);Benzamide, N-[2,3-dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxy-;FQWDVNSBYDXPIO-CQSZACIVSA-N;N-[2,3-dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide;CS-2243;BRPF1 bromodomain inhibitor GS6853;GSK-6853;GSK 6853
45 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- Ambeed
- ApexBio Technology
- AvaChem
- Biosynth
- BroadPharm
- Cayman Chemical
- ChemScene
- DC Chemicals
- Sigma-Aldrich
- Tocris
- TRC
Package
- 10mM*1mLinDMSO
- 1mg
- 5
- 2mg
- 5mg
- 10mg
- 25
- 25mg
- 50mg
- 100mg
- 200mg
- 250mg
- 1G
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98%
- Packaging1mg
- Price$24
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98%
- Packaging2mg
- Price$29
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98%
- Packaging5mg
- Price$41
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98%
- Packaging10mg
- Price$67
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98
- Packaging25mg
- Price$115
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98
- Packaging50mg
- Price$179
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98
- Packaging100mg
- Price$276
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00ABPJ
- Product descriptionN-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98
- Packaging200mg
- Price$383
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberM15357
- Product descriptionGSK6853 98%
- Packaging100MG
- Price$220
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberM15357
- Product descriptionGSK6853 98%
- Packaging1G
- Price$1100
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product number5421EG
- Product descriptionN-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide
- Packaging50mg
- Price$640
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number5421EG
- Product descriptionN-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide
- Packaging10mg
- Price$218
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA181180
- Product descriptionGSK6853 98+%
- Packaging50mg
- Price$145
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA181180
- Product descriptionGSK6853 98+%
- Packaging25mg
- Price$111
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA181180
- Product descriptionGSK6853 98+%
- Packaging10mg
- Price$85
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA181180
- Product descriptionGSK6853 98+%
- Packaging5mg
- Price$65
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98% | 1mg | $24 | 2026-05-28 | Buy |
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98% | 2mg | $29 | 2026-05-28 | Buy |
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98% | 5mg | $41 | 2026-05-28 | Buy |
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98% | 10mg | $67 | 2026-05-28 | Buy |
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98 | 25mg | $115 | 2026-05-28 | Buy |
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98 | 50mg | $179 | 2026-05-28 | Buy |
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98 | 100mg | $276 | 2026-05-28 | Buy |
| aablocks | AA00ABPJ | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide 98 | 200mg | $383 | 2026-05-28 | Buy |
| ACHEMBLOCK | M15357 | GSK6853 98% | 100MG | $220 | 2026-05-27 | Buy |
| ACHEMBLOCK | M15357 | GSK6853 98% | 1G | $1100 | 2026-05-27 | Buy |
| AK Scientific | 5421EG | N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide | 50mg | $640 | 2021-12-16 | Buy |
| AK Scientific | 5421EG | N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide | 10mg | $218 | 2021-12-16 | Buy |
| Ambeed | A181180 | GSK6853 98+% | 50mg | $145 | 2021-12-16 | Buy |
| Ambeed | A181180 | GSK6853 98+% | 25mg | $111 | 2021-12-16 | Buy |
| Ambeed | A181180 | GSK6853 98+% | 10mg | $85 | 2021-12-16 | Buy |
| Ambeed | A181180 | GSK6853 98+% | 5mg | $65 | 2021-12-16 | Buy |
Properties
Boiling point :545.9±50.0 °C(Predicted)
Density :1.247±0.06 g/cm3(Predicted)
storage temp. :Sealed in dry,Store in freezer, under -20°C
solubility :Soluble in DMSO (25 mg/ml); ethanol (25 mg/ml)
form :solid
pka :13.03±0.20(Predicted)
color :White
optical activity :[α]/D -45 to -55°, c =0.3 in methanol
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
InChIKey :FQWDVNSBYDXPIO-CQSZACIVSA-N
SMILES :O=C1N(C)C2=CC(N3CCNC[C@H]3C)=C(NC(C4=C(OC)C=CC=C4)=O)C=C2N1C
Density :1.247±0.06 g/cm3(Predicted)
storage temp. :Sealed in dry,Store in freezer, under -20°C
solubility :Soluble in DMSO (25 mg/ml); ethanol (25 mg/ml)
form :solid
pka :13.03±0.20(Predicted)
color :White
optical activity :[α]/D -45 to -55°, c =0.3 in methanol
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
InChIKey :FQWDVNSBYDXPIO-CQSZACIVSA-N
SMILES :O=C1N(C)C2=CC(N3CCNC[C@H]3C)=C(NC(C4=C(OC)C=CC=C4)=O)C=C2N1C
Safety Information
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Description
GSK6853 (1910124-24-1) is a very potent (pIC50 = 8.6 vs full length protein, 7.7 in cellular assays) inhibitor of Bromodomain and PHD Finger-containing 1 (BRPF1). It displayed >1600-fold selectivity over other bromodomains.Related product price
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Suppliers and manufacturers
Shanghai Boyle Chemical Co., Ltd.
BOC Sciences
MedChemexpress LLC
Bide Pharmatech Ltd.
Shanghai Lollane Biological Technology Co.,Ltd.
Shanghaizehan biopharma technology co., Ltd.
Shanghai YuanYe Biotechnology Co., Ltd.
Shanghai Chaolan Chemical Technology Center
Beijing Solarbio Science & Tecnology Co., Ltd.
Amadis Chemical Company Limited