S1RA
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- $81 - $2691.1
- Product name: S1RA
- CAS: 878141-96-9
- MF: C20H23N3O2
- MW: 337.42
- EINECS:
- MDL Number:MFCD25976945
- Synonyms:S1RA;4-(2-(5-METHYL-1-(NAPHTHALEN-2-YL)-1H-PYRAZOL-3-YLOXY)ETHYL)MORPHOLINE. HCL;4-[2-[[5-Methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine;4-[2-[[5-Methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine S1RA;S1RA 4-[2-[[5-Methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine;S1RA, >=98%;S1RA, 878141-96-9;4-(2-((5-Methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yl)oxy)ethyl)morpholine
17 prices
Selected condition：
Brand
- ApexBio Technology
- Biorbyt Ltd
- Cayman Chemical
- Chemenu
- Crysdot
- DC Chemicals
- Sigma-Aldrich
Package
- 500μg
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 1g
- 1 unit
- 10mM(in 1mL DMSO)
- 250mg
- 1000mg
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging5mg
- Price$280
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging10mM(in 1mL DMSO)
- Price$300
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging10mg
- Price$400
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB1179
- Product descriptionS1RA
- Packaging50mg
- Price$1200
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181123
- Product descriptionS1RA >98%
- Packaging100mg
- Price$765
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181123
- Product descriptionS1RA >98%
- Packaging250mg
- Price$1504.5
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181123
- Product descriptionS1RA >98%
- Packaging1000mg
- Price$2691.1
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging500μg
- Price$81
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging1mg
- Price$152
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging5mg
- Price$435
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number16279
- Product descriptionS1RA ≥98%
- Packaging10mg
- Price$711
- Updated2024-03-01
- Buy
- ManufacturerChemenu
- Product numberCM141471
- Product description4-(2-((5-Methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yl)oxy)ethyl)morpholine 98%
- Packaging100mg
- Price$884
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31000448
- Product descriptionS1RA 98+%
- Packaging25mg
- Price$378
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31000448
- Product descriptionS1RA 98+%
- Packaging100mg
- Price$945
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7274
- Product descriptionS1RA >98%
- Packaging100mg
- Price$500
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7274
- Product descriptionS1RA >98%
- Packaging1g
- Price$1800
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| ApexBio Technology | B1179 | S1RA | 5mg | $280 | 2021-12-16 | Buy |
| ApexBio Technology | B1179 | S1RA | 10mM(in 1mL DMSO) | $300 | 2021-12-16 | Buy |
| ApexBio Technology | B1179 | S1RA | 10mg | $400 | 2021-12-16 | Buy |
| ApexBio Technology | B1179 | S1RA | 50mg | $1200 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181123 | S1RA >98% | 100mg | $765 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181123 | S1RA >98% | 250mg | $1504.5 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181123 | S1RA >98% | 1000mg | $2691.1 | 2021-12-16 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 500μg | $81 | 2024-03-01 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 1mg | $152 | 2024-03-01 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 5mg | $435 | 2024-03-01 | Buy |
| Cayman Chemical | 16279 | S1RA ≥98% | 10mg | $711 | 2024-03-01 | Buy |
| Chemenu | CM141471 | 4-(2-((5-Methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yl)oxy)ethyl)morpholine 98% | 100mg | $884 | 2021-12-16 | Buy |
| Crysdot | CD31000448 | S1RA 98+% | 25mg | $378 | 2021-12-16 | Buy |
| Crysdot | CD31000448 | S1RA 98+% | 100mg | $945 | 2021-12-16 | Buy |
| DC Chemicals | DC7274 | S1RA >98% | 100mg | $500 | 2021-12-16 | Buy |
| DC Chemicals | DC7274 | S1RA >98% | 1g | $1800 | 2021-12-16 | Buy |
Properties
Boiling point :528.1±50.0 °C(Predicted)
Density :1.21±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :≥10.35 mg/mL in DMSO; ≥12.23 mg/mL in EtOH; ≥56.1 mg/mL in H2O
form :solid
pka :6.15±0.10(Predicted)
color :Off-white to yellow
Density :1.21±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :≥10.35 mg/mL in DMSO; ≥12.23 mg/mL in EtOH; ≥56.1 mg/mL in H2O
form :solid
pka :6.15±0.10(Predicted)
color :Off-white to yellow
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
The sigma-1 (σ1) receptor is an intracellular, non-opioid receptor that is abundantly expressed in the central nervous system as well as peripherally. S1RA is a potent, selective antagonist of σ1 receptors (Ki = 17 nM) that weakly binds σ2 receptors (Ki = 9,300 nM). It is active in vivo, dose-dependently inhibiting neuropathic pain in several animal models, including formalin-induced nociception and capsaicin-induced mechanical hypersensitivity. S1RA enhances peripheral μ-opioid analgesia without affecting opioid-induced constipation.Suppliers and manufacturers
ATK CHEMICAL COMPANY LIMITED
Zhejiang J&C Biological Technology Co.,Limited
InvivoChem
ShenZhen Trendseen Biological Technology Co.,Ltd.
Wuhan Topule Biopharmaceutical Co., Ltd
Zibo Hangyu Biotechnology Development Co., Ltd
HANGZHOU LEAP CHEM CO., LTD.
Aladdin Scientific
Amadis Chemical Company Limited
